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1 . Academic Journal
Dynamic Profiling and Binding Affinity Prediction of NBTI Antibacterials against DNA Gyrase Enzyme by Multidimensional Machine Learning and Molecular Dynamics Simulations
저자
by
Maja Kokot
;
Nikola Minovski
.
소스
ACS Omega, Vol 9, Iss 16, Pp 18278-18295 (2024)
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4 . Academic Journal
Exploring Alternative Pathways to Target Bacterial Type II Topoisomerases Using NBTI Antibacterials: Beyond Halogen-Bonding Interactions
저자
by
Maja Kokot
;
Doroteja Novak
;
Irena Zdovc
;
Marko Anderluh
;
Martina Hrast
, et al.
소스
Antibiotics, Vol 12, Iss 5, p 930 (2023)
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7 . Academic Journal
A Fine-Tuned Lipophilicity/Hydrophilicity Ratio Governs Antibacterial Potency and Selectivity of Bifurcated Halogen Bond-Forming NBTIs
저자
by
Anja Kolarič
;
Maja Kokot
;
Martina Hrast
;
Matjaž Weiss
;
Irena Zdovc
, et al.
소스
Antibiotics, Vol 10, Iss 7, p 862 (2021)
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7 .
Amide containing NBTI antibacterials with reduced hERG inhibition, retained antimicrobial activity against gram-positive bacteria and in vivo efficacy
저자
by
Maja Kokot
;
Matjaž Weiss
;
Irena Zdovc
;
Lidija Senerovic
;
Natasa Radakovic
, et al.
소스
European journal of medicinal chemistry, str. 1-13 : Ilustr., Vol. 250, 2023
COBISS-ID: 25429760
European journal of medicinal chemistry, vol. 115160, no. 250, pp. 1-13, 2023.
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7 .
Diminishing hERG inhibitory activity of aminopiperidine-naphthyridine linked NBTI antibacterials by structural and physicochemical optimizations
저자
by
Maja Kokot
;
Matjaž Weiss
;
Irena Zdovc
;
Marko Anderluh
;
Martina Hrast
, et al.
소스
Bioorganic chemistry, 14 str. : Ilustr., Vol. 128, 2022
COBISS-ID: 25099008
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7 .
The structural features of novel bacterial topoisomerase inhibitors that define their activity on topoisomerase IV
저자
by
Maja Kokot
;
Marko Anderluh
;
Martina Hrast
;
Nikola Minovski
.
소스
Journal of medicinal chemistry, vol. 65, no. 9, 2022.
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6 .
A Fine-Tuned Lipophilicity/Hydrophilicity Ratio Governs Antibacterial Potency and Selectivity of Bifurcated Halogen Bond-Forming NBTIs
저자
by
Irena Zdovc
;
Matjaž Weiss
;
Marko Anderluh
;
Anja Kolarič
;
Simon Žakelj
, et al.
소스
Antibiotics
Volume 10
Issue 7
Antibiotics, 30 str. : Ilustr., tabele, Vol. 10, no. 7, art. 862, 2021
COBISS-ID: 522975769
Antibiotics, Vol 10, Iss 862, p 862 (2021)
Antibiotics, vol. 10, no. 7, 862, 2021.
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7 .
Structurally Optimized Potent Dual-Targeting NBTI Antibacterials with an Enhanced Bifurcated Halogen-Bonding Propensity
저자
by
Irena Zdovc
;
Nikola Minovski
;
Martina Hrast
;
Matjaž Weiss
;
Maja Kokot
, et al.
소스
ACS Medicinal Chemistry Letters
ACS medicinal chemistry letters, vol. 12, no. 9, pp. 1478-1485, 2021.
ACS Medicinal Chemistry Letters, str. 1478-1485 : Ilustr., Vol. 12, iss. 9, 2021
COBISS-ID: 2959217
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