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1 . Academic Journal
Scaffold-hopping identifies furano[2,3-d]pyrimidine amides as potent Notum inhibitors
저자
by
Atkinson, Benjamin N.
;
Steadman, David
;
Mahy, William
;
Zhao, Yuguang
;
Sipthorp, James
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 February 2020 30(3)
Full Text (ScienceDirect)
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7 . Academic Journal
Structural Analysis and Development of Notum Fragment Screening Hits.
저자
by
Zhao, Yuguang
;
Mahy, William
;
Willis, Nicky J.
;
Woodward, Hannah L.
;
Steadman, David
, et al.
소스
ACS Chemical Neuroscience; 7/6/2022, Vol. 13 Issue 3, p2060-2077, 18p
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7 . Academic Journal
Bimodal regulation of axonal transport by the GDNF-RET signalling axis in healthy and diseased motor neurons.
저자
by
Rhymes, Elena R.
;
Tosolini, Andrew P.
;
Fellows, Alexander D.
;
Mahy, William
;
McDonald, Neil Q.
, et al.
소스
Cell Death & Disease; Jul2022, Vol. 13 Issue 7, p1-14, 14p
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7 . Academic Journal
Design of a Potent, Selective, and Brain-Penetrant Inhibitor of Wnt-Deactivating Enzyme Notum by Optimization of a Crystallographic Fragment Hit.
저자
by
Willis, Nicky J.
;
Mahy, William
;
Sipthorp, James
;
Zhao, Yuguang
;
Woodward, Hannah L.
, et al.
소스
Journal of Medicinal Chemistry; 5/26/2022, Vol. 65 Issue 10, p7212-7230, 19p
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7 . Dissertation/ Thesis
Catalytic synthesis and modification of heterocycles
저자
by
Mahy, William
;
Frost, Christopher
;
Plucinski, Pawel
.
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5 . Academic Journal
5‑Phenyl-1,3,4-oxadiazol-2(3H)‑ones Are Potent Inhibitors of Notum Carboxylesterase Activity Identified by the Optimization of a Crystallographic Fragment Screening Hit.
저자
by
Mahy, William
;
Willis, Nicky J.
;
Zhao, Yuguang
;
Woodward, Hannah L.
;
Svensson, Fredrik
, et al.
소스
Journal of Medicinal Chemistry; 11/12/2020, Vol. 63 Issue 21, p12942-12956, 15p
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7 . Academic Journal
Screening of a Custom-Designed Acid Fragment Library Identifies 1‑Phenylpyrroles and 1‑Phenylpyrrolidines as Inhibitors of Notum Carboxylesterase Activity.
저자
by
Mahy, William
;
Patel, Mikesh
;
Steadman, David
;
Woodward, Hannah L.
;
Atkinson, Benjamin N.
, et al.
소스
Journal of Medicinal Chemistry; 9/10/2020, Vol. 63 Issue 17, p9464-9483, 20p
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7 . Periodical
The medicinal chemistry of mitochondrial dysfunction: a critical overview of efforts to modulate mitochondrial healthElectronic supplementary information (ESI) available. See DOI: 10.1039/d1md00113b
저자
by
Lee, Maximillian Taro William
;
Mahy, William
;
Rackham, Mark David
.
소스
MedChemComm; 2021, Vol. 12 Issue: 8 p1281-1311, 31p
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5 . Academic Journal
A Highly Regioselective Palladium-Catalyzed O,S Rearrangement of Cyclic Thiocarbonates.
저자
by
Mahy, William
;
Cabezas‐Hayes, Sinéad
;
Kociok‐Köhn, Gabriele
;
Frost, Christopher G.
.
소스
European Journal of Organic Chemistry
. 11/24/2017, Vol. 2017 Issue 43, p6441-6444. 4p.
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6 . Academic Journal
Copper Catalyzed Assembly of N-Aryloxazolidinones: Synthesis of Linezolid, Tedizolid, and Rivaroxaban.
저자
by
Mahy, William
;
Leitch, Jamie A.
;
Frost, Christopher G.
.
소스
European Journal of Organic Chemistry
. Mar2016, Vol. 2016 Issue 7, p1305-1313. 9p.
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