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1 .
Abstract 4114: Evaluation of AU-18069, a novel small molecule CBP/p300 bromodomain inhibitor for the treatment of cancers
저자
by
Chandrasekhar Abbineni
;
Saravanan Thiyagarajan
;
Aravind A B
;
Amit A Dhudashiya
;
Sivapriya Marappan
, et al.
소스
Cancer Research
. 82:4114-4114
Full Text (AACR)
Web of Science
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7 .
Selective PPARδ Modulators Improve Mitochondrial Function: Potential Treatment for Duchenne Muscular Dystrophy (DMD)
저자
by
Bharat Lagu
;
Eric L. Bell
;
Effie Tozzo
;
Nirbhay Kumar Tiwari
;
Andrew Basinski
, et al.
소스
ACS Medicinal Chemistry Letters
. 9:935-940
Open Access (OpenAIRE)
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7 .
Highly selective peroxisome proliferator-activated receptor δ (PPARδ) modulator demonstrates improved safety profile compared to GW501516
저자
by
Ross Fredenburg
;
Matthew M. Goddeeris
;
Shekar Chellur
;
Ramesh S. Senaiar
;
Bharat Lagu
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 28:533-536
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7 .
Abstract 1143: Evaluation of AU-18069, a novel small molecule CBP/p300 bromodomain inhibitor for the treatment of cancers
저자
by
Samiulla D S
;
Shekar Chelur
;
Pathange Hemasankar
;
Mikko Myllymäki
;
Kavitha Nellore
, et al.
소스
Cancer Research
. 81:1143-1143
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7 . Academic Journal
LRRK2 phosphorylates moesin at threonine-558: characterization of how Parkinson's disease mutants affect kinase activity.
저자
by
Mahaboobi Jaleel
;
R. Jeremy Nichols
;
Maria Deak
;
David G. Campbell
;
Frank Gillardon
, et al.
소스
Biochemical Journal
. 2007, Vol. 405 Issue 0, p307-317. 11p.
Web of Science
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7 .
Correction to 'Selective PPARδ Modulators Improve Mitochondrial Function: Potential Treatment for Duchenne Muscular Dystrophy (DMD)'
저자
by
Mahaboobi Jaleel
;
Matthew M. Goddeeris
;
Ramesh S. Senaiar
;
Peter Dwyer
;
Eric L. Bell
, et al.
소스
Open Access (OpenAIRE)
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7 .
Abstract 1754: First in class orally bioavailable BETBRD degraders
저자
by
Avainash Kumar
;
Olli Törmäkangas
;
Susanta Samajdar
;
AB Aravind
;
Suraj Tgore
, et al.
소스
Cancer Research
. 80:1754-1754
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7 .
Structure-guided discovery of 2-aryl/pyridin-2-yl-1H-indole derivatives as potent and selective hepsin inhibitors
저자
by
Karthikeyan Narasingapuram Arumugam
;
Jwala Nagaraj
;
DS Samiulla
;
Murali Ramachandra
;
Rajendra K. Palakurthy
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 25:5309-5314
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7 .
Novel highly selective inhibitors of ubiquitin specific protease 30 (USP30) accelerate mitophagy
저자
by
Bharat Lagu
;
Michael Webb
;
Pranab Maiti
;
Arthur F. Kluge
;
Jyoti Malhotra
, et al.
소스
Bioorganicmedicinal chemistry letters
. 28(15)
Full Text (ScienceDirect)
Scopus
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7 .
Novel highly selective peroxisome proliferator-activated receptor δ (PPARδ) modulators with pharmacokinetic properties suitable for once-daily oral dosing
저자
by
Sunil Kumar Panigrahi
;
Effie Tozzo
;
Narasimha Rao Krishnamurthy
;
Taisuke Takahashi
;
Mahaboobi Jaleel
, et al.
소스
Bioorganicmedicinal chemistry letters
. 27(23)
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