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1 . Academic Journal
Identification of RP-6685, an Orally Bioavailable Compound that Inhibits the DNA Polymerase Activity of Polθ.
저자
by
Bubenik, Monica
;
Mader, Pavel
;
Mochirian, Philippe
;
Vallée, Fréderic
;
Clark, Jillian
, et al.
소스
Journal of Medicinal Chemistry; 10/13/2022, Vol. 65 Issue 19, p13198-13215, 18p
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7 . Academic Journal
Discovery and Structural Characterization of Small Molecule Binders of the Human CTLH E3 Ligase Subunit GID4.
저자
by
Chana, Chetan K.
;
Maisonneuve, Pierre
;
Posternak, Ganna
;
Grinberg, Nicolas G.A.
;
Poirson, Juline
, et al.
소스
Journal of Medicinal Chemistry; 10/13/2022, Vol. 65 Issue 19, p12725-12746, 22p
Full Text (ACS)
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7 . Academic Journal
Discovery of an Orally Bioavailable and Selective PKMYT1 Inhibitor, RP-6306.
저자
by
Szychowski, Janek
;
Papp, Robert
;
Dietrich, Evelyne
;
Liu, Bingcan
;
Vallée, Frédéric
, et al.
소스
Journal of Medicinal Chemistry; 8/11/2022, Vol. 65 Issue 15, p10251-10284, 34p
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7 . Periodical
Functional characterization of a PROTAC directed against BRAF mutant V600E
저자
by
Posternak, Ganna
;
Tang, Xiaojing
;
Maisonneuve, Pierre
;
Jin, Ting
;
Lavoie, Hugo
, et al.
소스
Nature Chemical Biology; November 2020, Vol. 16 Issue: 11 p1170-1178, 9p
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7 . Academic Journal
Identification and characterization of the first fragment hits for SETDB1 Tudor domain.
저자
by
Mader, Pavel
;
Mendoza-Sanchez, Rodrigo
;
Iqbal, Aman
;
Dong, Aiping
;
Dobrovetsky, Elena
, et al.
소스
Bioorganic & Medicinal Chemistry
. Sep2019, Vol. 27 Issue 17, p3866-3878. 13p.
Full Text (ScienceDirect)
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7 . Academic Journal
Crystal structure of native α‐l‐rhamnosidase from Aspergillus terreus.
저자
by
Pachl, Petr
;
Škerlová, Jana
;
Šimčíková, Daniela
;
Kotik, Michael
;
Křenková, Alena
, et al.
소스
Acta Crystallographica: Section D, Structural Biology
. Nov2018, Vol. 74 Issue 11, p1078-1084. 7p.
Find it @ DONGA
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7 . Academic Journal
Carborane-Based Carbonic Anhydrase Inhibitors: Insight into CAII/CAIX Specificity from a High-Resolution Crystal Structure, Modeling, and Quantum Chemical Calculations.
저자
by
Mader, Pavel
;
Pecina, Adam
;
Cígler, Petr
;
Lepšík, Martin
;
Šícha, Václav
, et al.
소스
BioMed Research International
. 2014, Vol. 2014, p1-9. 9p.
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7 . Academic Journal
QM/MM CalculationsReveal the Different Nature ofthe Interaction of Two Carborane-Based Sulfamide Inhibitors of HumanCarbonic Anhydrase II.
저자
by
Pecina, Adam
;
Lepšík, Martin
;
Řezáč, Jan
;
Brynda, Jiří
;
Mader, Pavel
, et al.
소스
Journal of Physical Chemistry B
. Dec2013, Vol. 117 Issue 50, p16096-16104. 9p.
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7 . Academic Journal
Carborane-Based Carbonic Anhydrase Inhibitors.
저자
by
Brynda, Jiří
;
Mader, Pavel
;
Šícha, Václav
;
Fábry, Milan
;
Poncová, Kristýna
, et al.
소스
Angewandte Chemie
. Dec2013, Vol. 125 Issue 51, p14005-14008. 4p.
Full Text (Wiley)
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7 . Periodical
Identification of a Fragment-like Small Molecule Ligand for the Methyl-lysine Binding Protein, 53BP1
저자
by
Perfetti, Michael T.
;
Baughman, Brandi M.
;
Dickson, Bradley M.
;
Mu, Yunxiang
;
Cui, Gaofeng
, et al.
소스
ACS Chemical Biology; April 2015, Vol. 10 Issue: 4 p1072-1081, 10p
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