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1 . Academic Journal
Discovery of the 1,7-diazacarbazole class of inhibitors of checkpoint kinase 1
저자
by
Gazzard, Lewis
;
Appleton, Brent
;
Chapman, Kerry
;
Chen, Huifen
;
Clark, Kevin
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 December 2014 24(24):5704-5709
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7 . Periodical
Discovery and Preclinical Characterization of BIIB091, a Reversible, Selective BTK Inhibitor for the Treatment of Multiple Sclerosis
저자
by
Hopkins, Brian T.
;
Bame, Eris
;
Bajrami, Bekim
;
Black, Cheryl
;
Bohnert, Tonika
, et al.
소스
Journal of Medicinal Chemistry; January 2022, Vol. 65 Issue: 2 p1206-1224, 19p
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7 . Academic Journal
Design, Synthesis, and Biological Investigation of Thailanstatin A and Spliceostatin D Analogues Containing Tetrahydropyran, Tetrahydrooxazine, and Fluorinated Structural Motifs.
저자
by
Nicolaou, K. C.
;
Rekula, Santhosh Reddy
;
Kumar, S. Mothish
;
Podilapu, Ananda Rao
;
Matuszak, Ryan P.
, et al.
소스
Journal of Organic Chemistry; 2/5/2021, Vol. 86 Issue 3, p2499-2521, 23p
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7 . Periodical
Design, Synthesis, and Biological Evaluation of Tubulysin Analogues, Linker-Drugs, and Antibody–Drug Conjugates, Insights into Structure–Activity Relationships, and Tubulysin–Tubulin Binding Derived from X-ray Crystallographic Analysis
저자
by
Nicolaou, K. C.
;
Pan, Saiyong
;
Pulukuri, Kiran K.
;
Ye, Qiuji
;
Rigol, Stephan
, et al.
소스
The Journal of Organic Chemistry; February 2021, Vol. 86 Issue: 4 p3377-3421, 45p
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7 . Academic Journal
Non-oxime pyrazole based inhibitors of B-Raf kinase
저자
by
Newhouse, Bradley J.
;
Hansen, Joshua D.
;
Grina, Jonas
;
Welch, Mike
;
Topalov, George
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(11):3488-3492
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7 . Academic Journal
Non-oxime inhibitors of B-Raf V600E kinase
저자
by
Ren, Li
;
Wenglowsky, Steve
;
Miknis, Greg
;
Rast, Bryson
;
Buckmelter, Alex J.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(4):1243-1247
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7 . Academic Journal
The Discovery of furo[2,3- c]pyridine-based indanone oximes as potent and selective B-Raf inhibitors
저자
by
Buckmelter, Alex J.
;
Ren, Li
;
Laird, Ellen R.
;
Rast, Bryson
;
Miknis, Greg
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(4):1248-1252
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7 . Periodical
Total Synthesis and Biological Evaluation of Tiancimycins A and B, Yangpumicin A, and Related Anthraquinone-Fused Enediyne Antitumor Antibiotics
저자
by
Nicolaou, K. C.
;
Das, Dipendu
;
Lu, Yong
;
Rout, Subhrajit
;
Pitsinos, Emmanuel N.
, et al.
소스
Journal of the American Chemical Society; February 2020, Vol. 142 Issue: 5 p2549-2561, 13p
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7 . Academic Journal
Potent and selective pyrazole-based inhibitors of B-Raf kinase
저자
by
Hansen, Joshua D.
;
Grina, Jonas
;
Newhouse, Brad
;
Welch, Mike
;
Topalov, George
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2008 18(16):4692-4695
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7 . Academic Journal
Mitigation of opioid off-target effects and identification of structural drivers of opioid receptor engagement for BACE-1 small molecule inhibitors.
저자
by
Diaz, Dolores
;
Dambach, Donna
;
Siu, Michael
;
Hunt, Kevin
;
Thomas, Allen
, et al.
소스
Toxicology Mechanisms & Methods
. Jul2015, Vol. 25 Issue 6, p478-486. 9p. 1 Color Photograph, 2 Diagrams, 5 Charts, 2 Graphs.
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