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1 . Academic Journal
The discovery of novel 5,6,5- and 5,5,6-tricyclic pyrrolidines as potent and selective DPP-4 inhibitors
저자
by
Cox, Jason M.
;
Chu, Hong D.
;
Kuethe, Jeffrey T.
;
Gao, Ying-Duo
;
Scapin, Giovanna
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 June 2016 26(11):2622-2626
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7 . Academic Journal
Structure–activity-relationship of amide and sulfonamide analogs of omarigliptin
저자
by
Chen, Ping
;
Feng, Dennis
;
Qian, Xiaoxia
;
Apgar, James
;
Wilkening, Robert
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 December 2015 25(24):5767-5771
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7 . Academic Journal
A novel benzazepinone sodium channel blocker with oral efficacy in a rat model of neuropathic pain
저자
by
Hoyt, Scott B.
;
London, Clare
;
Abbadie, Catherine
;
Felix, John P.
;
Garcia, Maria L.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 June 2013 23(12):3640-3645
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7 . Academic Journal
Pyridinesulfonylureas and pyridinesulfonamides as selective bombesin receptor subtype-3 (BRS-3) agonists
저자
by
Lo, Michael M.-C.
;
Chobanian, Harry R.
;
Palyha, Oksana
;
Kan, Yanqing
;
Kelly, Theresa M.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(7):2040-2043
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7 . Academic Journal
Synthesis and evaluation of [(1 R)-1-amino-2-(2,5-difluorophenyl)ethyl]cyclohexanes and 4-[(1 R)-1-amino-2-(2,5-difluorophenyl)ethyl]piperidines as DPP-4 inhibitors
저자
by
Chen, Ping
;
Caldwell, Charles G.
;
Ashton, Wallace
;
Wu, Joseph K.
;
He, Huaibing
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(6):1880-1886
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7 . Academic Journal
A potent and selective indole N-type calcium channel (Ca v2.2) blocker for the treatment of pain
저자
by
Tyagarajan, Sriram
;
Chakravarty, Prasun K.
;
Park, Min
;
Zhou, Bishan
;
Herrington, James B.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(2):869-873
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7 . Academic Journal
Discovery of a novel class of biphenyl pyrazole sodium channel blockers for treatment of neuropathic pain
저자
by
Tyagarajan, Sriram
;
Chakravarty, Prasun K.
;
Zhou, Bishan
;
Taylor, Brett
;
Eid, Ronsar
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(24):7479-7482
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7 . Academic Journal
Aminopiperidine-fused imidazoles as dipeptidyl peptidase-IV inhibitors
저자
by
Edmondson, Scott D.
;
Mastracchio, Anthony
;
Cox, Jason M.
;
Eiermann, George J.
;
He, Huaibing
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 August 2009 19(15):4097-4101
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7 . Academic Journal
Discovery of isoxazole voltage gated sodium channel blockers for treatment of chronic pain
저자
by
Shao, Pengcheng P.
;
Ye, Feng
;
Weber, Ann E.
;
Li, Xiaohua
;
Lyons, Kathryn A.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2009 19(18):5334-5338
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7 . Academic Journal
Discovery of a novel class of isoxazoline voltage gated sodium channel blockers
저자
by
Shao, Pengcheng P.
;
Ye, Feng
;
Weber, Ann E.
;
Li, Xiaohua
;
Lyons, Kathryn A.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2009 19(18):5329-5333
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