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1 . Academic Journal
Discovery of 5-Chloro-N2-[(1S)-1-(5-fluoropyrimidin-2-yl)ethyl]-N4-(5-methyl-1H-pyrazol-3-yl)pyrimidine-2,4-diamine (AZD1480) as a Novel Inhibitor of the Jak/Stat Pathway.
저자
by
Stephanos Ioannidis
;
Michelle L. Lamb
;
Tao Wang
;
Lynsie Almeida
;
Michael H. Block
, et al.
소스
Journal of Medicinal Chemistry
. Jan2011, Vol. 54 Issue 1, p262-276. 15p.
Full Text (ACS)
Web of Science
Scopus
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7 .
Synthesis of Novel Hydroxymethyl-Substituted Fused Heterocycles
저자
by
Laksmaiah Gingipalli
;
Jane E. Moore
;
Rosemary A. Croft
;
Barlaam Bernard Christophe
;
Janet Hawkins
, et al.
소스
Synthesis
. 48:1226-1234
Web of Science
Scopus
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7 .
Discovery of AZ0108, an orally bioavailable phthalazinone PARP inhibitor that blocks centrosome clustering
저자
by
Nancy Su
;
Xin Wang
;
Keith Mikule
;
Lynsie Almeida
;
Xiaolan Zheng
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 25:5743-5747
Web of Science
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7 .
Discovery of 1-Methyl-1H-imidazole Derivatives as Potent Jak2 Inhibitors
저자
by
Tina Howard
;
Jie Shi
;
Kirsten Bell
;
Jon Read
;
Dennis Huszar
, et al.
소스
Journal of Medicinal Chemistry
. 57:144-158
Web of Science
Scopus
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7 .
Discovery of pyrazol-3-ylamino pyrazines as novel JAK2 inhibitors
저자
by
Michelle Lamb
;
Geraldine Bebernitz
;
Marat Alimzhanov
;
Michael Zinda
;
Davies Audrey
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 19:6524-6528
Web of Science
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7 .
Discovery of a novel class of 2-ureido thiophene carboxamide checkpoint kinase inhibitors
저자
by
Candice Horn
;
Martin Pass
;
James W. Janetka
;
Kevin Daly
;
Nicholas John Newcombe
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 18:4242-4248
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7 .
Pyrimidinone nicotinamide mimetics as selective tankyrase and wnt pathway inhibitors suitable for in vivo pharmacology
저자
by
Graeme R. Robb
;
Lynsie Almeida
;
Rosemary A. Croft
;
Jian Huang
;
Haiyun Wang
, et al.
소스
ACS medicinal chemistry letters
. 6(3)
Open Access (OpenAIRE)
Scopus
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7 .
Discovery of checkpoint kinase inhibitor (S)-5-(3-fluorophenyl)-N-(piperidin-3-yl)-3-ureidothiophene-2-carboxamide (AZD7762) by structure-based design and optimization of thiophenecarboxamide ureas
저자
by
Siân Rowsell
;
Shannon Ready
;
James W. Janetka
;
Dongfang Liu
;
Paul Lyne
, et al.
소스
Journal of medicinal chemistry
. 55(11)
Scopus
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7 .
Discovery of 5-chloro-N2-[(1S)-1-(5-fluoropyrimidin-2-yl)ethyl]-N4-(5-methyl-1H-pyrazol-3-yl)pyrimidine-2,4-diamine (AZD1480) as a novel inhibitor of the Jak/Stat pathway
저자
by
Hai-Jun Zhang
;
Tina Howard
;
Isabelle Green
;
Marat Alimzhanov
;
Minwei Ye
, et al.
소스
Journal of medicinal chemistry
. 54(1)
Scopus
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7 .
Replacement of pyrazol-3-yl amine hinge binder with thiazol-2-yl amine: Discovery of potent and selective JAK2 inhibitors
저자
by
Geraldine Bebernitz
;
Marat Alimzhanov
;
Guan Huiping
;
Bo Peng
;
Lynsie Almeida
, et al.
소스
Bioorganicmedicinal chemistry letters
. 20(5)
Full Text (ScienceDirect)
Scopus
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