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1 . Academic Journal
Garbage in, garbage out: how reliable training data improved a virtual screening approach against SARS-CoV-2 MPro
저자
by
Santiago M. Ruatta
;
Denis N. Prada Gori
;
Martín Fló Díaz
;
Franca Lorenzelli
;
Karen Perelmuter
, et al.
소스
Frontiers in Pharmacology, Vol 14 (2023)
Open Access (DOAJ)
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7 . Academic Journal
Drug repurposing screening validated by experimental assays identifies two clinical drugs targeting SARS-CoV-2 main protease
저자
by
Denis N. Prada Gori
;
Santiago Ruatta
;
Martín Fló
;
Lucas N. Alberca
;
Carolina L. Bellera
, et al.
소스
Frontiers in Drug Discovery, Vol 2 (2023)
Open Access (DOAJ)
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7 . Academic Journal
LIDeB Tools: A Latin American resource of freely available, open-source cheminformatics apps
저자
by
Denis N. Prada Gori
;
Lucas N. Alberca
;
Santiago Rodriguez
;
Juan I. Alice
;
Manuel A. Llanos
, et al.
소스
Artificial Intelligence in the Life Sciences, Vol 2, Iss , Pp 100049- (2022)
Full Text (ScienceDirect)
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Full Text (ScienceDirect O/A)
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7 . Academic Journal
In silico Guided Drug Repurposing: Discovery of New Competitive and Non-competitive Inhibitors of Falcipain-2
저자
by
Lucas N. Alberca
;
Sara R. Chuguransky
;
Cora L. Álvarez
;
Alan Talevi
;
Emir Salas-Sarduy
.
소스
Frontiers in Chemistry, Vol 7 (2019)
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7 . Academic Journal
Cascade Ligand- and Structure-Based Virtual Screening to Identify New Trypanocidal Compounds Inhibiting Putrescine Uptake
저자
by
Lucas N. Alberca
;
María L. Sbaraglini
;
Juan F. Morales
;
Roque Dietrich
;
María D. Ruiz
, et al.
소스
Frontiers in Cellular and Infection Microbiology, Vol 8 (2018)
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7 .
Making the most effective use of available computational methods for drug repositioning
저자
by
Denis N. Prada Gori
;
Lucas N. Alberca
;
Alan Talevi
.
소스
Expert Opinion on Drug Discovery
. 18:495-503
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5 .
A combined ligand and target-based virtual screening strategy to repurpose drugs as putrescine uptake inhibitors with trypanocidal activity
저자
by
Manuel A. Llanos
;
Lucas N. Alberca
;
María D. Ruiz
;
María L. Sbaraglini
;
Cristian Miranda
, et al.
소스
Journal of Computer-Aided Molecular Design
. 37:75-90
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7 .
iRaPCA and SOMoC: Development and Validation of Web Applications for New Approaches for the Clustering of Small Molecules
저자
by
Denis N. Prada Gori
;
Manuel A. Llanos
;
Carolina L. Bellera
;
Alan Talevi
;
Lucas N. Alberca
.
소스
Journal of Chemical Information and Modeling
. 62:2987-2998
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7 .
Tetracycline Derivatives Inhibit Plasmodial Cysteine Protease Falcipain-2 through Binding to a Distal Allosteric Site
저자
by
Jorge Enrique Hernández González
;
Lucas N. Alberca
;
Yordanka Masforrol González
;
Osvaldo Reyes Acosta
;
Alan Talevi
, et al.
소스
Scopus
Repositório Institucional da UNESP
Universidade Estadual Paulista (UNESP)
instacron:UNESP
Open Access (OpenAIRE)
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7 .
Machine Learning Search of Novel Selective NaV1.2 and NaV1.6 Inhibitors as Potential Treatment Against Dravet Syndrome
저자
by
Maximiliano Fallico
;
Lucas N. Alberca
;
Denis N. Prada Gori
;
Luciana Gavernet
;
Alan Talevi
.
소스
Communications in Computer and Information Science ISBN: 9783031084423
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