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1 . Academic Journal
Dose-dependent effects of GAT107, a novel allosteric agonist-positive allosteric modulator (ago-PAM) for the α7 nicotinic cholinergic receptor: a BOLD phMRI and connectivity study on awake rats
저자
by
Brittany M. Brems
;
Erin E. Sullivan
;
Jenna G. Connolly
;
Jingchun Zhang
;
Arnold Chang
, et al.
소스
Frontiers in Neuroscience, Vol 17 (2023)
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7 . Academic Journal
Use of a Molecular Switch Probe to Activate or Inhibit GIRK1 Heteromers In Silico Reveals a Novel Gating Mechanism
저자
by
Dimitrios Gazgalis
;
Lucas Cantwell
;
Yu Xu
;
Ganesh A. Thakur
;
Meng Cui
, et al.
소스
International Journal of Molecular Sciences, Vol 23, Iss 18, p 10820 (2022)
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7 .
Development of novel subtype-selective modulators of heteromeric girk channels
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by
Lucas Cantwell
.
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3 .
Negative allosteric modulation of CBsub1/subcannabinoid receptor signaling suppresses opioid-mediated reward
저자
by
Vishakh Iyer
;
Claudia Rangel-Barajas
;
Taylor J. Woodward
;
Abhijit Kulkarni
;
Lucas Cantwell
, et al.
소스
Pharmacol Res
Open Access (OpenAIRE)
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7 .
Allosterically Potentiated α7 Nicotinic Acetylcholine Receptors: Reduced Calcium Permeability and Current-Independent Control of Intracellular Calcium
저자
by
Douglas R. Miller
;
Roger L. Papke
;
Sumanta Garai
;
Lucas Cantwell
;
Ganesh A. Thakur
, et al.
소스
Mol Pharmacol
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7 .
The small molecule GAT1508 activates brain-specific GIRK1/2 channel heteromers and facilitates conditioned fear extinction in rodents
저자
by
Yuchen Yang
;
Lucas Cantwell
;
Diomedes E. Logothetis
;
Erik T. Dustrude
;
Leigh D. Plant
, et al.
소스
J Biol Chem
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7 .
Heteromeric Neuronal Nicotinic Acetylcholine Receptors with Mutant β Subunits Acquire Sensitivity to α7-Selective Positive Allosteric Modulators
저자
by
Khalil A. Abboud
;
Clare Stokes
;
Nicole A. Horenstein
;
Abhijit R. Kulkarni
;
Roger L. Papke
, et al.
소스
J Pharmacol Exp Ther
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7 .
A benzopyran with antiarrhythmic activity is an inhibitor of Kir3.1-containing potassium channels
저자
by
Haozhou Tan
;
Diomedes E. Logothetis
;
Ganesh A. Thakur
;
Mengmeng Chang
;
Said EI-Haou
, et al.
소스
The Journal of Biological Chemistry
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7 .
Kir Channel Molecular Physiology, Pharmacology, and Therapeutic Implications
저자
by
Lucas Cantwell
;
Andrew Zorn
;
Meng Cui
;
Diomedes E. Logothetis
.
소스
Pharmacology of Potassium Channels ISBN: 9783030840518
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6 .
Molecular Mechanism of the Potent Benzopyran-G1 Blocker of Heteromeric G-Protein Gated Potassium Channels
저자
by
Sami F. Noujaim
;
Keman Xu
;
Haozhou Tan
;
Diomedes E. Logothetis
;
Said EI-Haou
, et al.
소스
Biophysical Journal
. 120:203a
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