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1 . Academic Journal
Benzimidazolone as potent chymase inhibitor: Modulation of reactive metabolite formation in the hydrophobic (P 1) region
저자
by
Lo, Ho Yin
;
Nemoto, Peter A.
;
Kim, Jin Mi
;
Hao, Ming-Hong
;
Qian, Kevin C.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(15):4533-4539
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7 . Academic Journal
Substituted pyrazoles as novel sEH antagonist: Investigation of key binding interactions within the catalytic domain
저자
by
Lo, Ho Yin
;
Man, Chuk C.
;
Fleck, Roman W.
;
Farrow, Neil A.
;
Ingraham, Richard H.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 November 2010 20(22):6379-6383
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7 . Academic Journal
2-Aminobenzimidazoles as potent ITK antagonists: trans-stilbene-like moieties targeting the kinase specificity pocket
저자
by
Lo, Ho Yin
;
Bentzien, Jörg
;
Fleck, Roman W.
;
Pullen, Steven S.
;
Khine, Hnin Hnin
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 December 2008 18(23):6218-6221
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7 . Academic Journal
2-Aminobenzimidazoles as potent ITK antagonists: de novo design of a pyrrole system targeting additional hydrogen bonding interaction
저자
by
Lo, Ho Yin
;
Bentzien, Jörg
;
White, Andre
;
Man, Chuk C.
;
Fleck, Roman W.
, et al.
소스
In
Tetrahedron Letters
2008 49(51):7337-7340
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7 . Academic Journal
Discovery, SAR and X-ray structure of 1 H-benzimidazole-5-carboxylic acid cyclohexyl-methyl-amides as inhibitors of inducible T-cell kinase (Itk)
저자
by
Moriarty, Kevin J.
;
Takahashi, Hidenori
;
Pullen, Steven S.
;
Khine, Hnin Hnin
;
Sallati, Rosemarie H.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2008 18(20):5545-5549
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7 . Academic Journal
Corrigendum to “Discovery, SAR and X-ray structure of 1 H-benzimidazole-5-carboxylic acid cyclohexyl-methyl-amides as inhibitors of inducible T-cell kinase (Itk)” [Bioorg. Med. Chem. Lett. 18 (2008) 5545–5549]
저자
by
Moriarty, Kevin J.
;
Takahashi, Hidenori
;
Pullen, Steven S.
;
Khine, Hnin Hnin
;
Sallati, Rosemarie H.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2009 19(6):1835-1835
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7 . Academic Journal
Benzimidazolone as potent chymase inhibitor: Modulation of reactive metabolite formation in the hydrophobic (P
1
) region
저자
by
Lo, Ho Yin
;
Nemoto, Peter A.
;
Kim, Jin Mi
;
Hao, Ming-Hong
;
Qian, Kevin C.
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. Aug2011, Vol. 21 Issue 15, p4533-4539. 7p.
Full Text (ScienceDirect)
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7 . Periodical
Itk inhibitors: a patent review
저자
by
Lo, Ho Yin
.
소스
Expert Opinion on Therapeutic Patents; January 2010, Vol. 20 Issue: 4 p459-469, 11p
Web of Science
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3 . Academic Journal
Synthesis, SAR, and Series Evolution of Novel Oxadiazole-Containing 5-Lipoxygenase Activating Protein Inhibitors: Discovery of 2-[4-(3-{(R)-1-[4-(2-Amino-pyrimidin-5-yl)-phenyl]-1-cyclopropyl-ethyl}-[1,2,4]oxadiazol-5-yl)-pyrazol-1-yl]-N,N-dimethyl-acetamide (BI 665915)
저자
by
Takahashi, Hidenori
;
Riether, Doris
;
Bartolozzi, Alessandra
;
Bosanac, Todd
;
Berger, Valentina
, et al.
소스
JOURNAL OF MEDICINAL CHEMISTRY
; FEB 26 2015, 58 4, p1669-p1690, 22p.
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7 . Patent
저자
by
Bartolozzi, Alessandra
;
Chen, Zhidong
;
Dines, Jonathon Alan
;
Lo, Ho Yin
;
Loke, Pui Leng
, et al.
소스
Open Access (USPTO)
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