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1 . Academic Journal
Large Scale Meta-Analysis of Fragment-Based Screening Campaigns: Privileged Fragments and Complementary Technologies
저자
by
Kutchukian, Peter S.
;
Wassermann, Anne Mai
;
Lindvall, Mika K.
;
Wright, S. Kirk
;
Ottl, Johannes
, et al.
소스
In
SLAS Discovery
June 2015 20(5):588-596
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7 . Academic Journal
Novel γ-turn mimetics with a reinforced hydrogen bond
저자
by
Lindvall, Mika K.
;
Rissanen, Kari
;
Hakala, Juha M.L.
;
Koskinen, Ari M.P.
.
소스
In
Tetrahedron Letters
1999 40(41):7427-7430
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6 . Academic Journal
Fragment-Based Drug Discovery of Inhibitors of Phosphopantetheine Adenylyltransferase from Gram-Negative Bacteria.
저자
by
Moreau, Robert J.
;
Skepper, Colin K.
;
Appleton, Brent A.
;
Blechschmidt, Anke
;
Balibar, Carl J.
, et al.
소스
Journal of Medicinal Chemistry
. 4/26/2018, Vol. 61 Issue 8, p3309-3324. 16p.
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7 . Academic Journal
Regiochemical observations on the lithiation of 1,2,4-trichlorobenzene and reaction with DMF and oxamide electrophiles in THF
저자
by
Burton, Andrew J.
;
Cardwell, Kevin S.
;
Fuchter, Matthew J.
;
Lindvall, Mika K.
;
Patel, Rajnikant
, et al.
소스
In
Tetrahedron Letters
2003 44(30):5653-5656
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7 . Academic Journal
Inside the Mind of a Medicinal Chemist: The Role of Human Bias in Compound Prioritization during Drug Discovery.
저자
by
Kutchukian, Peter S.
;
Vasilyeva, Nadya Y.
;
Xu, Jordan
;
Lindvall, Mika K.
;
Dillon, Michael P.
, et al.
소스
PLoS ONE
. Nov2012, Vol. 7 Issue 11, Special section p1-18. 18p.
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7 . Academic Journal
Origins of stereoselectivity in the Corey-Chaykovsky reaction. Insights from quantum chemistry.
저자
by
Lindvall, Mika K.
;
Koskinen, Ari M.P.
.
소스
Journal of Organic Chemistry
. 06/25/99, Vol. 64 Issue 13, p4598. 11p. 8 Diagrams, 8 Charts, 2 Graphs.
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4 . Periodical
The Application of Quantitative Analytical Constructs for Chemistry Optimization, Monomer Rehearsal and Reactivity Prediction in Solid Phase Library Synthesis
저자
by
Parr, Nigel J.
;
McKeown, Stephen C.
;
Lindvall, Mika K.
;
Lorthioir, Olivier E.
;
Congreve, Miles S.
, et al.
소스
Letters in Organic Chemistry; January 01, 2004, Vol. 1 Issue: 1 p87-92, 6p
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7 . Periodical
The Binding Mode of Calyculin A to Protein Phosphatase-1
저자
by
Lindvall, Mika K.
;
Pihko, Petri M.
;
Koskinen, Ari M.P.
.
소스
Journal of Biological Chemistry; September 1997, Vol. 272 Issue: 37 p23312-23316, 5p
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5 . Academic Journal
Identification of N-(4-((1R,3S,5S)-3-Amino-5-methylcyclohexyl)pyridin-3-yl)-6-(2,6-difluorophenyl)-5-fluoropicolinamide (PIM447), a Potent and Selective Proviral Insertion Site of Moloney Murine Leukemia (PIM) 1, 2, and 3 Kinase Inhibitor in Clinical Trials for Hematological Malignancies
저자
by
Burger, Matthew T.
;
Nishiguchi, Gisele
;
Han, Wooseok
;
Lan, Jiong
;
Simmons, Robert
, et al.
소스
JOURNAL OF MEDICINAL CHEMISTRY
; NOV 12 2015, 58 21, p8373-p8386, 14p.
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7 . Academic Journal
Optimization of a Dibenzodiazepine Hit to a Potent and Selective Allosteric PAK1 Inhibitor
저자
by
Karpov, Alexei S.
;
Amiri, Payman
;
Bellamacina, Cornelia
;
Bellance, Marie-Helene
;
Breitenstein, Werner
, et al.
소스
ACS MEDICINAL CHEMISTRY LETTERS
; JUL 2015, 6 7, p776-p781, 6p.
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