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1 . Academic Journal
PETRANHA: Phase 1/2 study of AZD5305 + novel hormonal agents in patients with metastatic prostate cancer–Interim safety and pharmacokinetic results.
저자
by
Azad, Arun
;
Voskoboynik, Mark
;
Joshua, Anthony M.
;
Weickhardt, Andrew James
;
Sankey, Peter
, et al.
소스
Journal of Clinical Oncology; 2024 Supplement 4, Vol. 42, p123-123, 235p
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7 . Academic Journal
Inhibition of Bromodomain Proteins Enhances Oncolytic HAdVC5 Replication and Efficacy in Pancreatic Ductal Adenocarcinoma (PDAC) Models.
저자
by
Miao, Tizong
;
Symonds, Alistair
;
Hickman, Oliver J.
;
Wu, Dongsheng
;
Wang, Ping
, et al.
소스
International Journal of Molecular Sciences
. Jan2024, Vol. 25 Issue 2, p1265. 21p.
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7 . Academic Journal
Tumour selective targeting of cell cycle kinases for cancer treatment
저자
by
Aarts, Marieke
;
Linardopoulos, Spiros
;
Turner, Nicholas C
.
소스
In
Current Opinion in Pharmacology
August 2013 13(4):529-535
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5 . Academic Journal
PPM1D gene amplification and overexpression in breast cancer: a qRT-PCR and chromogenic in situ hybridization study
저자
by
Lambros, Maryou B
;
Natrajan, Rachael
;
Geyer, Felipe C
;
Lopez-Garcia, Maria A
;
Dedes, Konstantin J
, et al.
소스
In
Modern Pathology
October 2010 23(10):1334-1345
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7 . Academic Journal
High-Throughput Screening Assay for Identification of Small Molecule Inhibitors of Aurora2/STK15 Kinase
저자
by
Sun, Chongbo
;
Newbatt, Yvette
;
Douglas, Leon
;
Workman, Paul
;
Aherne, Wynne
, et al.
소스
In
SLAS Discovery
August 2004 9(5):391-397
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7 . Academic Journal
7-(Pyrazol-4-yl)-3H-imidazo[4,5-b]pyridine-based derivatives for kinase inhibition: Co-crystallisation studies with Aurora-A reveal distinct differences in the orientation of the pyrazole N1-substituent
저자
by
Bavetsias, Vassilios
;
Pérez-Fuertes, Yolanda
;
McIntyre, Patrick J.
;
Atrash, Butrus
;
Kosmopoulou, Magda
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 October 2015 25(19):4203-4209
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7 . Academic Journal
CCT245718, a dual FLT3/Aurora A inhibitor overcomes D835Y-mediated resistance to FLT3 inhibitors in acute myeloid leukaemia cells.
저자
by
Tariq, Muhammad Usama
;
Furqan, Muhammad
;
Parveen, Hira
;
Ullah, Rahim
;
Muddassar, Muhammad
, et al.
소스
British Journal of Cancer
. Sep2021, Vol. 125 Issue 7, p966-974. 9p.
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7 . Academic Journal
Targeting the PPM1D phenotype; 2,4-bisarylthiazoles cause highly selective apoptosis in PPM1D amplified cell-lines
저자
by
Cheeseman, Matthew D.
;
Faisal, Amir
;
Rayter, Sydonia
;
Barbeau, Olivier R.
;
Kalusa, Andrew
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 August 2014 24(15):3469-3474
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7 . Academic Journal
Adaptation of the plasma inhibitory activity assay to detect Aurora, ABL and FLT3 kinase inhibition by AT9283 in pediatric leukemia
저자
by
Podesta, Jennifer E.
;
Sugar, Richard
;
Squires, Matt
;
Linardopoulos, Spiros
;
Pearson, Andrew D.J.
, et al.
소스
In
Leukemia Research
2011 35(9):1273-1275
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7 . Academic Journal
Structure-based design of imidazo[1,2- a]pyrazine derivatives as selective inhibitors of Aurora-A kinase in cells
저자
by
Bouloc, Nathalie
;
Large, Jonathan M.
;
Kosmopoulou, Magda
;
Sun, Chongbo
;
Faisal, Amir
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(20):5988-5993
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