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1 . Academic Journal
Phase 1 and preclinical profiling of ESM‐HDAC391, a myeloid‐targeted histone deacetylase inhibitor, shows enhanced pharmacology and monocytopaenia.
저자
by
Furze, Rebecca C.
;
Molnar, Judit
;
Parr, Nigel J.
;
Ahmad, Faiz
;
Henry, Yvette
, et al.
소스
British Journal of Clinical Pharmacology
. Dec2022, Vol. 88 Issue 12, p5238-5256. 19p.
Web of Science
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7 . Academic Journal
Fr481 CARBOXYLESTERASE-1 ASSISTED TARGETING OF HDAC INHIBITOR TO MONONUCLEAR MYELOID CELLS ATTENUATES COLON INFLAMMATION IN T CELL TRANSFER COLITIS MURINE MODEL.
저자
by
Elfiky, Ahmed
;
Hageman, Ishtu
;
Van Hamersveld, Patricia
;
Welting, Olaf
;
Verhoeff, Jan
, et al.
소스
In
Gastroenterology
May 2021 160(6) Supplement:S
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7 . Academic Journal
Optimisation of a novel series of potent and orally bioavailable azanaphthyridine SYK inhibitors
저자
by
Garton, Neil S.
;
Barker, Michael D.
;
Davis, Rob P.
;
Douault, Clement
;
Hooper-Greenhill, Edward
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 October 2016 26(19):4606-4612
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7 . Academic Journal
Mo1104 MONONUCLEAR MYELOID CELL TARGETED HISTONE DEACETYLASE (HDAC) INHIBITOR DEMONSTRATES POTENT ACTIVITY IN MONOCYTES AND IMPAIRS COLON MONOCYTES TO MACROPHAGE DIFFERENTIATION DURING ACUTE DSS COLITIS.
저자
by
Elfiky, Ahmed
;
Ghiboub, Mohammed
;
Hamersveld, Patricia H.P.van
;
Welting, Olaf
;
van den berg, iris
, et al.
소스
In
Gastroenterology
May 2020 158(6) Supplement 1:S
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7 . Academic Journal
Preclinical models of arthritis for studying immunotherapy and immune tolerance.
저자
by
Meehan, Gavin R.
;
Thomas, Ranjeny
;
Al Khabouri, Shaima
;
Wehr, Pascale
;
Hilkens, Catharien M. U.
, et al.
소스
Annals of the Rheumatic Diseases; Oct2021, Vol. 80 Issue 10, p1268-1277, 10p
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7 . Academic Journal
BRD4 methylation by the methyltransferase SETD6 regulates selective transcription to control mRNA translation.
저자
by
Vershinin, Zlata
;
Feldman, Michal
;
Werner, Thilo
;
Estrella Weil, Lital
;
Kublanovsky, Margarita
, et al.
소스
Science Advances
. 5/26/2021, Vol. 7 Issue 22, p1-13. 13p.
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7 . Academic Journal
Novel Insights Into Rheumatoid Arthritis Through Characterization of Concordant Changes in DNA Methylation and Gene Expression in Synovial Biopsies of Patients With Differing Numbers of Swollen Joints.
저자
by
Li Yim, Andrew Y. F.
;
Ferrero, Enrico
;
Maratou, Klio
;
Lewis, Huw D.
;
Royal, George
, et al.
소스
Frontiers in Immunology; 4/22/2021, Vol. 11, pN.PAG-N.PAG, 15p
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7 . Academic Journal
Targeting Histone Deacetylases in Myeloid Cells Inhibits Their Maturation and Inflammatory Function With Limited Effects on Atherosclerosis.
저자
by
Luque-Martin, Rosario
;
Van den Bossche, Jan
;
Furze, Rebecca C.
;
Neele, Annette E.
;
van der Velden, Saskia
, et al.
소스
Frontiers in Pharmacology; 10/29/2019, Vol. 10, p1-14, 14p
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7 . Academic Journal
Discovery of GSK143, a highly potent, selective and orally efficacious spleen tyrosine kinase inhibitor
저자
by
Liddle, John
;
Atkinson, Francis L.
;
Barker, Michael D.
;
Carter, Paul S.
;
Curtis, Neil R.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2011 21(20):6188-6194
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7 . Academic Journal
3-Substituted gem-cyclohexane sulfone based γ-secretase inhibitors for Alzheimer’s disease: Conformational analysis and biological activity
저자
by
Jelley, Richard A.
;
Elliott, Jason
;
Gibson, Karl R.
;
Harrison, Timothy
;
Beher, Dirk
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2006 16(14):3839-3842
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