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1 . Academic Journal
Optimization and biological evaluation of thiazole-bis-amide inverse agonists of RORγt
저자
by
Gege, Christian
;
Albers, Michael
;
Kinzel, Olaf
;
Kleymann, Gerald
;
Schlüter, Thomas
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 June 2020 30(12)
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7 . Academic Journal
Novel potent and selective α vβ 3/α vβ 5 integrin dual antagonists with reduced binding affinity for human serum albumin
저자
by
Raboisson, Pierre
;
Manthey, Carl L.
;
Chaikin, Margery
;
Lattanze, Jennifer
;
Crysler, Carl
, et al.
소스
In
European Journal of Medicinal Chemistry
2006 41(7):847-861
Full Text (ScienceDirect)
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7 . Academic Journal
3-Substituted Quinolines as RORγt Inverse Agonists
저자
by
Tanis, Virginia M.
;
Venkatesan, Hariharan
;
Cummings, Maxwell D.
;
Albers, Michael
;
Kent Barbay, J.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 June 2019 29(12):1463-1470
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7 . Academic Journal
A functional radioreceptor assay of alpha-V-beta-3 (α vβ 3) inhibitors in plasma: Application as an ex vivo pharmacodynamic model
저자
by
Chaikin, Margery A.
;
Marugan, Júan José
;
De Vries, Gerald W.
;
Baciu, Peter
;
Edelman, Jeffrey
, et al.
소스
In
Journal of Biochemical and Biophysical Methods
2005 65(2):107-120
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7 . Academic Journal
Identification and biological evaluation of thiazole-based inverse agonists of RORγt
저자
by
Gege, Christian
;
Cummings, Maxwell D.
;
Albers, Michael
;
Kinzel, Olaf
;
Kleymann, Gerald
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 May 2018 28(9):1446-1455
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7 . Academic Journal
6-Substituted quinolines as RORγt inverse agonists
저자
by
Barbay, J. Kent
;
Cummings, Maxwell D.
;
Abad, Marta
;
Castro, Glenda
;
Kreutter, Kevin D.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 December 2017 27(23):5277-5283
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7 . Academic Journal
Identification and structure activity relationships of quinoline tertiary alcohol modulators of RORγt
저자
by
Kummer, David A.
;
Cummings, Maxwell D.
;
Abad, Marta
;
Barbay, Joseph
;
Castro, Glenda
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 May 2017 27(9):2047-2057
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7 . Academic Journal
Substituted thieno[2,3-d]pyrimidines as adenosine A2A receptor antagonists
저자
by
Shook, Brian C.
;
Chakravarty, Devraj
;
Barbay, J. Kent
;
Wang, Aihua
;
Leonard, Kristi
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 May 2013 23(9):2688-2691
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7 . Academic Journal
Design and synthesis of polyethylene glycol-modified biphenylsulfonyl-thiophene-carboxamidine inhibitors of the complement component C1s
저자
by
Subasinghe, Nalin L.
;
Khalil, Ehab
;
Travins, Jeremy M.
;
Ali, Farah
;
Ballentine, Shelley K.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 August 2012 22(16):5303-5307
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7 . Academic Journal
Optimization of arylindenopyrimidines as potent adenosine A 2A/A 1 antagonists
저자
by
Shook, Brian C.
;
Rassnick, Stefanie
;
Chakravarty, Devraj
;
Wallace, Nathaniel
;
Ault, Mark
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(9):2868-2871
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