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1 . Academic Journal
Novel LC/MS/MS and High-Throughput Mass Spectrometric Assays for Monoacylglycerol Acyltransferase Inhibitors
저자
by
Qi, Jenson
;
Masucci, John A.
;
Lang, Wensheng
;
Connelly, Margery A.
;
Caldwell, Gary W.
, et al.
소스
In
SLAS Discovery
April 2017 22(4):433-439
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7 . Academic Journal
5,5-Difluoro- and 5-Fluoro-5-methyl-hexose-based C-Glucosides as potent and orally bioavailable SGLT1 and SGLT2 dual inhibitors
저자
by
Xu, Guozhang
;
Du, Fuyong
;
Kuo, Gee-Hong
;
Xu, June Zhi
;
Liang, Yin
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 September 2020 30(17)
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7 . Academic Journal
Design, synthesis and biological evaluation of (2S,3R,4R,5S,6R)-5-fluoro-6-(hydroxymethyl)-2-aryltetrahydro-2H-pyran-3,4-diols as potent and orally active SGLT dual inhibitors
저자
by
Xu, Guozhang
;
Gaul, Michael D.
;
Kuo, Gee-Hong
;
Du, Fuyong
;
Xu, June Zhi
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 November 2018 28(21):3446-3453
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7 . Academic Journal
Synthesis and biological evaluation of novel macrocyclic bis-7-azaindolylmaleimides as potent and highly selective glycogen synthase kinase-3β (GSK-3β) inhibitors
저자
by
Shen, Lan
;
Prouty, Catherine
;
Conway, Bruce R.
;
Westover, Lori
;
Xu, Jun Z.
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 March 2004 12(5):1239-1255
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7 . Academic Journal
Design, synthesis, and biological evaluation of novel 7-azaindolyl-heteroaryl-maleimides as potent and selective glycogen synthase kinase-3β (GSK-3β) inhibitors
저자
by
O'Neill, David J.
;
Shen, Lan
;
Prouty, Catherine
;
Conway, Bruce R.
;
Westover, Lori
, et al.
소스
In
Bioorganic & Medicinal Chemistry
2004 12(12):3167-3185
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7 . Academic Journal
Synthesis and biological evaluation of benzocyclobutane-C-glycosides as potent and orally active SGLT1/SGLT2 dual inhibitors
저자
by
Kuo, Gee-Hong
;
Gaul, Micheal D.
;
Liang, Yin
;
Xu, June Z.
;
Du, Fuyong
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 April 2018 28(7):1182-1187
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7 . Academic Journal
4-Bicyclic heteroaryl-piperidine derivatives as potent, orally bioavailable stearoyl-CoA desaturase-1 (SCD1) inhibitors: Part 2. Pyridazine-based analogs
저자
by
Yang, Shyh-Ming
;
Tang, Yuting
;
Rano, Thomas
;
Lu, Huajun
;
Kuo, Gee-Hong
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 March 2014 24(5):1437-1441
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7 . Academic Journal
4-Bicyclic heteroaryl-piperidine derivatives as potent, orally bioavailable Stearoyl-CoA desaturase-1 (SCD1) inhibitors. Part 1: Urea-based analogs
저자
by
Yang, Shyh-Ming
;
Tang, Yuting
;
Zhang, Rui
;
Lu, Huajun
;
Kuo, Gee-Hong
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 December 2013 23(24):6773-6776
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7 . Academic Journal
Optimization of a pyrazole hit from FBDD into a novel series of indazoles as ketohexokinase inhibitors
저자
by
Zhang, Xuqing
;
Song, Fengbing
;
Kuo, Gee-Hong
;
Xiang, Amy
;
Gibbs, Alan C.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 August 2011 21(16):4762-4767
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7 . Academic Journal
Synthesis and discovery of 2,3-dihydro-3,8-diphenylbenzo[1,4]oxazines as a novel class of potent cholesteryl ester transfer protein inhibitors
저자
by
Wang, Aihua
;
Prouty, Catherine P.
;
Pelton, Patricia D.
;
Yong, Maria
;
Demarest, Keith T.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(4):1432-1435
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