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1 . Academic Journal
Discovery and SAR of JTE-151: A Novel RORγ Inhibitor for Clinical Development.
저자
by
Maeba, Takaki
;
Hirata, Kazuyuki
;
Kotoku, Masayuki
;
Seki, Noriyoshi
;
Maeda, Katsuya
, et al.
소스
Journal of Medicinal Chemistry; 1/25/2024, Vol. 67 Issue 2, p952-970, 19p
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7 . Academic Journal
Identification of Diketopiperazine-Containing 2‑Anilinobenzamides as Potent Sirtuin 2 (SIRT2)-Selective Inhibitors Targeting the "Selectivity Pocket", Substrate-Binding Site, and NAD
+
‑Binding Site.
저자
by
Mellini, Paolo
;
Itoh, Yukihiro
;
Elboray, Elghareeb E.
;
Tsumoto, Hiroki
;
Li, Ying
, et al.
소스
Journal of Medicinal Chemistry; 6/27/2019, Vol. 62 Issue 12, p5844-5862, 19p
Full Text (ACS)
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7 . Academic Journal
Discovery of Second Generation RORγ Inhibitors Composed of an Azole Scaffold.
저자
by
Kotoku, Masayuki
;
Maeba, Takaki
;
Fujioka, Shingo
;
Yokota, Masahiro
;
Seki, Noriyoshi
, et al.
소스
Journal of Medicinal Chemistry; 3/14/2019, Vol. 62 Issue 5, p2837-2842, 6p
Full Text (ACS)
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7 . Periodical
Identification of Diketopiperazine-Containing 2-Anilinobenzamides as Potent Sirtuin 2 (SIRT2)-Selective Inhibitors Targeting the “Selectivity Pocket”, Substrate-Binding Site, and NAD+-Binding Site
저자
by
Mellini, Paolo
;
Itoh, Yukihiro
;
Elboray, Elghareeb E.
;
Tsumoto, Hiroki
;
Li, Ying
, et al.
소스
Journal of Medicinal Chemistry; June 2019, Vol. 62 Issue: 12 p5844-5862, 19p
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7 . Academic Journal
Ternary complex of human RORγ ligand-binding domain, inverse agonist and SMRT peptide shows a unique mechanism of corepressor recruitment.
저자
by
Noguchi, Masato
;
Nomura, Akihiro
;
Murase, Ken
;
Doi, Satoki
;
Yamaguchi, Keishi
, et al.
소스
Genes to Cells
. Jun2017, Vol. 22 Issue 6, p535-551. 17p.
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7 . Academic Journal
Ternary crystal structure of human ROR gamma ligand-binding-domain, an inhibitor and corepressor peptide provides a new insight into corepressor interaction
저자
by
Noguchi, Masato
;
Nomura, Akihiro
;
Doi, Satoki
;
Yamaguchi, Keishi
;
Hirata, Kazuyuki
, et al.
소스
SCIENTIFIC REPORTS
; NOV 26 2018, 8 p17374 8p.
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7 . Academic Journal
A Study of C-F...M[sup +] Interaction: Alkali Metal Complexes of the Fluorine-Containing Cage...
저자
by
Takemura, Hiroyuki
;
Kon, Noriyoshi
;
Kotoku, Masayuki
;
Nakashima, Sachiko
;
Otsuka, Kazuhiro
, et al.
소스
Journal of Organic Chemistry
. 04/20/2001, Vol. 66 Issue 8, p2778. 6p. 5 Diagrams, 3 Charts, 5 Graphs.
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7 . Periodical
9-Fluoro-18-hydroxy-[3.3]metacyclophane: Synthesis and Estimation of a C−F···H−O Hydrogen Bond
저자
by
Takemura, Hiroyuki
;
Kotoku, Masayuki
;
Yasutake, Mikio
;
Shinmyozu, Teruo
.
소스
European Journal of Organic Chemistry; May 2004, Vol. 2004 Issue: 9 p2019-2024, 6p
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6 . Periodical
Identification of Potent and Selective Inhibitors of Fat Mass Obesity-Associated Protein Using a Fragment-Merging Approach
저자
by
Prakash, Muthuraj
;
Itoh, Yukihiro
;
Fujiwara, Yoshie
;
Takahashi, Yukari
;
Takada, Yuri
, et al.
소스
Journal of Medicinal Chemistry; 20210101, Issue: Preprints
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7 . Academic Journal
SAR Exploration Guided by LE and Fsp(3): Discovery of a Selective and Orally Efficacious ROR gamma Inhibitor
저자
by
Hirata, Kazuyuki
;
Kotoku, Masayuki
;
Seki, Noriyoshi
;
Maeba, Takaki
;
Maeda, Katsuya
, et al.
소스
ACS MEDICINAL CHEMISTRY LETTERS
; JAN 2016, 7 1, p23-p27, 5p.
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