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1 . Academic Journal
Novel potent and highly selective DDR1 inhibitors from integrated lead finding.
저자
by
Kuhn, Bernd
;
Ritter, Martin
;
Benz, Jörg
;
Kocer, Buelent
;
Sarie, Jérôme C.
, et al.
소스
Medicinal Chemistry Research; Jul2023, Vol. 32 Issue 7, p1400-1425, 26p
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7 . Academic Journal
Mitigation of reactive metabolite formation for a series of 3-amino-2-pyridone inhibitors of Bruton’s tyrosine kinase (BTK)
저자
by
Lou, Yan
;
Lopez, Francisco
;
Jiang, Yongying
;
Han, Xiaochun
;
Brotherton, Chris
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 February 2017 27(3):632-635
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7 . Academic Journal
Finding the perfect spot for fluorine: Improving potency up to 40-fold during a rational fluorine scan of a Bruton’s Tyrosine Kinase (BTK) inhibitor scaffold
저자
by
Lou, Yan
;
Sweeney, Zachary K.
;
Kuglstatter, Andreas
;
Davis, Dana
;
Goldstein, David M.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 January 2015 25(2):367-371
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7 . Academic Journal
Discovery of carmegliptin: A potent and long-acting dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes
저자
by
Mattei, Patrizio
;
Boehringer, Markus
;
Di Giorgio, Patrick
;
Fischer, Holger
;
Hennig, Michael
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(3):1109-1113
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7 . Academic Journal
DNA-Encoded Library-Derived DDR1 Inhibitor Prevents Fibrosis and Renal Function Loss in a Genetic Mouse Model of Alport Syndrome.
저자
by
Richter, Hans
;
Satz, Alexander L.
;
Bedoucha, Marc
;
Buettelmann, Bernd
;
Petersen, Ann C.
, et al.
소스
ACS Chemical Biology; Jan2019, Vol. 14 Issue 1, p37-49, 13p
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7 . Academic Journal
Discovery and Pre-Clinical Characterization of Third-Generation 4-H Heteroaryldihydropyrimidine (HAP) Analogues as Hepatitis B Virus (HBV) Capsid Inhibitors.
저자
by
Zongxing Qiu
;
Xianfeng Lin
;
Weixing Zhang
;
Mingwei Zhou
;
Lei Guo
, et al.
소스
Journal of Medicinal Chemistry
. 4/27/2017, Vol. 60 Issue 8, p3352-3371. 20p.
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7 . Academic Journal
Structure-Based Drug Designof RN486, a Potent andSelective Bruton’s Tyrosine Kinase (BTK) Inhibitor, for theTreatment of Rheumatoid Arthritis.
저자
by
Lou, Yan
;
Han, Xiaochun
;
Kuglstatter, Andreas
;
Kondru, Rama K.
;
Sweeney, Zachary K.
, et al.
소스
Journal of Medicinal Chemistry
. Jan2015, Vol. 58 Issue 1, p512-516. 5p.
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7 . Academic Journal
Discovery and Pre-Clinical Characterization of Third-Generation 4-H Heteroaryldihydropyrimidine (HAP) Analogues as Hepatitis B Virus (HBV) Capsid Inhibitors
저자
by
Qiu, Zongxing
;
Lin, Xianfeng
;
Zhang, Weixing
;
Zhou, Mingwei
;
Guo, Lei
, et al.
소스
JOURNAL OF MEDICINAL CHEMISTRY
; APR 27 2017, 60 8, p3352-p3371, 20p.
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7 .
Meteorological Conditions Related to the Onset of Spontaneous Pneumothorax
저자
by
Oezpolat, Berkant
;
Goezuebueyuek, Alper
;
Kocer, Buelent
;
Yazkan, Rasih
;
Dural, Koray
, et al.
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7 . Academic Journal
Complications of Tube Thoracostomy in 603 Patients
저자
by
Kocer, Buelent
;
Gulbahar, Gueltekin
;
Yildirim, Erkan
;
Dural, Koray
;
Sakinci, Uenal
.
소스
TURKIYE KLINIKLERI TIP BILIMLERI DERGISI
; JUN 2010, 30 3, p895-p899, 5p.
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