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1 . Academic Journal
Exploring the chemical space of orally bioavailable PROTACs
저자
by
Apprato, Giulia
;
Poongavanam, Vasanthanathan
;
Garcia Jimenez, Diego
;
Atilaw, Yoseph
;
Erdelyi, Mate
, et al.
소스
In
Drug Discovery Today
April 2024 29(4)
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7 . Academic Journal
Structure-based virtual screening discovers potent and selective adenosine A1 receptor antagonists
저자
by
Matricon, Pierre
;
Nguyen, Anh TN.
;
Vo, Duc Duy
;
Baltos, Jo-Anne
;
Jaiteh, Mariama
, et al.
소스
In
European Journal of Medicinal Chemistry
5 September 2023 257
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7 . Academic Journal
Predicting the Permeability of Macrocycles from Conformational Sampling – Limitations of Molecular Flexibility
저자
by
Poongavanam, Vasanthanathan
;
Atilaw, Yoseph
;
Ye, Sofie
;
Wieske, Lianne H.E.
;
Erdelyi, Mate
, et al.
소스
In
Journal of Pharmaceutical Sciences
January 2021 110(1):301-313
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7 . Academic Journal
Molecular chameleons in drug discovery.
저자
by
Poongavanam, Vasanthanathan
;
Wieske, Lianne H. E.
;
Peintner, Stefan
;
Erdélyi, Máté
;
Kihlberg, Jan
.
소스
Nature Reviews Chemistry; Jan2024, Vol. 8 Issue 1, p45-60, 16p
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7 . Academic Journal
Oral Druggable Space beyond the Rule of 5: Insights from Drugs and Clinical Candidates
저자
by
Doak, Bradley Croy
;
Over, Bjӧrn
;
Giordanetto, Fabrizio
;
Kihlberg, Jan
.
소스
In
Chemistry & Biology
18 September 2014 21(9):1115-1142
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6 . Academic Journal
Autoantibodies to Disease‐Related Proteins in Joints as Novel Biomarkers for the Diagnosis of Rheumatoid Arthritis.
저자
by
Lönnblom, Erik
;
Leu Agelii, Monica
;
Sareila, Outi
;
Cheng, Lei
;
Xu, Bingze
, et al.
소스
Arthritis & Rheumatology
. Jul2023, Vol. 75 Issue 7, p1110-1119. 10p.
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7 . Academic Journal
Hypothesis driven drug design: improving quality and effectiveness of the design-make-test-analyse cycle
저자
by
Plowright, Alleyn T.
;
Johnstone, Craig
;
Kihlberg, Jan
;
Pettersson, Jonas
;
Robb, Graeme
, et al.
소스
In
Drug Discovery Today
2012 17(1):56-62
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7 . Academic Journal
Therapy targeting antigen-specific T cells by a peptide-based tolerizing vaccine against autoimmune arthritis.
저자
by
Urbonaviciute, Vilma
;
Romero-Castillo, Laura
;
Bingze Xu
;
Huqiao Luo
;
Schneider, Nadine
, et al.
소스
Proceedings of the National Academy of Sciences of the United States of America
. 6/20/2023, Vol. 120 Issue 25, p1-10. 32p.
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7 . Academic Journal
Design of Drug Efficacy Guided by Free Energy Simulations of the β
2
‐Adrenoceptor.
저자
by
Panel, Nicolas
;
Vo, Duc Duy
;
Kahlous, Nour Aldin
;
Hübner, Harald
;
Tiedt, Stephanie
, et al.
소스
Angewandte Chemie
. 5/22/2023, Vol. 135 Issue 22, p1-10. 10p.
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7 . Academic Journal
Macrocycles in Drug DiscoveryLearning from the Past for the Future.
저자
by
Garcia Jimenez, Diego
;
Poongavanam, Vasanthanathan
;
Kihlberg, Jan
.
소스
Journal of Medicinal Chemistry; 4/27/2023, Vol. 66 Issue 8, p5377-5396, 20p
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