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1 . Academic Journal
Characterization of the mechanism of action of lanraplenib, a novel spleen tyrosine kinase inhibitor, in models of lupus nephritis
저자
by
Christopher W. Pohlmeyer
;
Ching Shang
;
Pei Han
;
Zhi-Hua Cui
;
Randall M. Jones
, et al.
소스
BMC Rheumatology, Vol 5, Iss 1, Pp 1-13 (2021)
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7 .
Small-molecule agents for the treatment of inflammatory bowel disease
저자
by
Sedillo Kassandra F
;
Leena Patel
;
Kevin S. Currie
.
소스
Bioorganic & Medicinal Chemistry Letters
. 29:2034-2041
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5 .
Effects of GS-9876, a novel spleen tyrosine kinase inhibitor, on platelet function and systemic hemostasis
저자
by
Emma Rousseau
;
Roy Bannister
;
Kevin S. Currie
;
Jiyun Kim
;
Astrid S. Clarke
, et al.
소스
Thrombosis Research
. 170:109-118
Full Text (Clinical Key)
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7 .
Discovery of Lanraplenib (GS-9876): A Once-Daily Spleen Tyrosine Kinase Inhibitor for Autoimmune Diseases
저자
by
Eric B. Lansdon
;
Helen Yu
;
Kropf Jeffrey E
;
Peter A. Blomgren
;
Jennifer R. Lo
, et al.
소스
ACS Med Chem Lett
Open Access (OpenAIRE)
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7 .
Discovery of Potent and Selective MTH1 Inhibitors for Oncology: Enabling Rapid Target (In)Validation
저자
by
Julie Farand
;
Jeffrey E. Kropf
;
Peter Blomgren
;
Jianjun Xu
;
Aaron C. Schmitt
, et al.
소스
ACS Med Chem Lett
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7 .
Discovery of Potent and Selective Tricyclic Inhibitors of Bruton’s Tyrosine Kinase with Improved Druglike Properties
저자
by
Steve Gallion
;
Jacob Z. Chen
;
Kropf Jeffrey E
;
Joseph W. Lubach
;
Pat Maciejewski
, et al.
소스
ACS Medicinal Chemistry Letters
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7 .
Discovery of highly potent and selective Bruton’s tyrosine kinase inhibitors: Pyridazinone analogs with improved metabolic stability
저자
by
James J. Crawford
;
Joseph W. Lubach
;
Peter Blomgren
;
Pat Maciejewski
;
Steve Gallion
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 26:575-579
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7 .
SAT0016 DEVELOPMENT OF FIBROBLAST-LIKE SYNOVIOCYTE ASSAYS FOR TARGET DISCOVERY IN RHEUMATOID ARTHRITIS
저자
by
V. Lira
;
G. Min-Oo
;
D. Ruelas
;
Kevin S. Currie
;
Helen Yu
, et al.
소스
Annals of the Rheumatic Diseases
. 79:938.1-938
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7 .
Potent and selective Bruton’s tyrosine kinase inhibitors: Discovery of GDC-0834
저자
by
Aaron C. Schmitt
;
Donna Dambach
;
Jen Macaluso
;
Kevin S. Currie
;
Xiaojing Wang
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 25(6):1333-1337
Full Text (ScienceDirect)
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7 .
Btk-specific inhibition blocks pathogenic plasma cell signatures and myeloid cell–associated damage in IFNα-driven lupus nephritis
저자
by
Laura DeForge
;
Eric Suto
;
Justin Lesch
;
Joseph W. Lubach
;
Arna Katewa
, et al.
소스
JCI Insight
. 2
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