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1 .
Discovery of Orally Bioavailable FGFR2/FGFR3 Dual Inhibitors via Structure-Guided Scaffold Repurposing Approach
저자
by
Minh H. Nguyen
;
Hai-Fen Ye
;
Yao Xu
;
Lisa Truong
;
April Horsey
, et al.
소스
ACS Medicinal Chemistry Letters
. 14:312-318
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7 .
Discovery of an Allosteric, Inactive Conformation-Selective Inhibitor of Full-Length HPK1 Utilizing a Kinase Cascade Assay
저자
by
Jorge Vialard
;
Kelly Federowicz
;
Geoff Struble
;
Weixue Wang
;
Samantha J Allen
, et al.
소스
Biochemistry
. 60(41)
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7 .
Lysine specific demethylase 1 inactivation enhances differentiation and promotes cytotoxic response when combined with all-trans retinoic acid in acute myeloid leukemia across subtypes
저자
by
Satyajit R. Rajapurkar
;
Kelly Federowicz
;
Rab K. Prinjha
;
Ashley M. Hughes
;
Elizabeth Thomas
, et al.
소스
Haematologica
Haematologica, 104(6)
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7 .
Generation and Validation of Intracellular Ubiquitin Variant Inhibitors for USP7 and USP10
저자
by
Li Liu
;
Dania Haddad
;
Sachdev S. Sidhu
;
Jingsong Yang
;
Dirk A. Heerding
, et al.
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7 .
Allosteric Wip1 phosphatase inhibition through flap-subdomain interaction
저자
by
Hong Zhang
;
Benjamin Schwartz
;
Michael D. Schaber
;
Mark A. Seefeld
;
Jon-Paul Jaworski
, et al.
소스
Nature Chemical Biology
. 10:181-187
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7 .
Long-Range Inhibitor-Induced Conformational Regulation of Human IRE1α Endoribonuclease Activity
저자
by
Sharon Sweitzer
;
Jeff Ralph
;
Maurice P. Deyoung
;
Angela Smallwood
;
William G. Bonnette
, et al.
소스
Molecular pharmacology
. 88(6)
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7 .
A DNA Hypomethylation Signature Predicts Antitumor Activity of LSD1 Inhibitors in SCLC
저자
by
Thau F. Ho
;
Yan Liu
;
Xinrong Tian
;
Patrick McDevitt
;
Michael Butticello
, et al.
소스
Cancer cell
. 28(1)
Full Text (ScienceDirect)
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7 .
Abstract 3513: Inhibition of LSD1 for the treatment of cancer
저자
by
Dominic Suarez
;
Glenn S. Van Aller
;
Jess Schneck
;
Kasparec Jiri
;
Kimberly N. Smitheman
, et al.
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Cancer Research
. 75:3513-3513
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7 .
Inhibition Of LSD1 As a Therapeutic Strategy For The Treatment Of Acute Myeloid Leukemia
저자
by
Jessica L. Schneck
;
Dominic Suarez
;
Peter J. Tummino
;
Scott A. Armstrong
;
Yan Liu
, et al.
소스
Blood
. 122:3964-3964
Full Text (ScienceDirect O/A)
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