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1 .
The Pharmacokinetics, Metabolism, and Clearance Mechanisms of Abrocitinib, a Selective Janus Kinase Inhibitor, in Humans
저자
by
Jonathan N. Bauman
;
Angela C. Doran
;
Amanda King-Ahmad
;
Raman Sharma
;
Gregory S. Walker
, et al.
소스
Drug Metabolism and Disposition
. 50:1106-1118
Web of Science
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7 .
Identification of Morpholino-2H-pyrido[3,2-b][1,4]oxazin-3(4H)-ones as Nonsteroidal Mineralocorticoid Antagonists
저자
by
Kentaro Futatsugi
;
Mary Ellen Banker
;
David W. Piotrowski
;
Kun Song
;
Michael Herr
, et al.
소스
Journal of Medicinal Chemistry
. 61:1086-1097
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7 .
P190 - The effect of CYP2C9 and CYP2C19 genotype on the pharmacokinetics of PF 04965842, A JAK1 inhibitor in clinical development
저자
by
Linda S. Wood
;
Jonathan N. Bauman
;
Jian Lin
;
Bimal Malhotra
;
Martin E. Dowty
, et al.
소스
Drug Metabolism and Pharmacokinetics
. 35:S80
Open Access (OpenAIRE)
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7 .
Undesired versus designed enzymatic cleavage of linkers for liver targeting
저자
by
Heather Eng
;
Jonathan N. Bauman
;
Robert L. Dow
;
M. G. Finn
;
Theunis C. Goosen
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 24:1144-1147
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7 .
Immune-Mediated Agranulocytosis Caused by the Cocaine Adulterant Levamisole: A Case for Reactive Metabolite(s) Involvement
저자
by
Steven Hansel
;
Jonathan N. Bauman
;
Amit S. Kalgutkar
;
Thomas S. McDonald
;
Yue Chen
, et al.
소스
Drug Metabolism and Disposition
. 40:1067-1075
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7 . Reference
Role of Metabolism in Toxicity of Drugs in Humans
저자
by
Amit S. Kalgutkar, author
;
Jonathan N. Bauman, author
;
Alexander V. Lyubimov, author
.
소스
Encyclopedia of Drug Metabolism and Interactions
. :1-26
Find it @ DONGA
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5 .
On-resin N-methylation of cyclic peptides for discovery of orally bioavailable scaffolds
저자
by
Spiros Liras
;
Cayla M. McEwen
;
Rushia A. Turner
;
David Price
;
Taha Rezai
, et al.
소스
Nature chemical biology
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7 .
Discovery Tactics To Mitigate Toxicity Risks Due to Reactive Metabolite Formation with 2-(2-Hydroxyaryl)-5-(trifluoromethyl)pyrido[4,3-d]pyrimidin-4(3H)-one Derivatives, Potent Calcium-Sensing Receptor Antagonists and Clinical Candidate(s) for the Treatment of Osteoporosis
저자
by
John R. Soglia
;
Hao Sun
;
Jonathan N. Bauman
;
Zhuang Miao
;
Jianke Li
, et al.
소스
Chemical Research in Toxicology
. 23:1115-1126
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7 .
The discovery of novel calcium sensing receptor negative allosteric modulators
저자
by
Gayatri Balan
;
Paul S. Humphries
;
David Price
;
Liuqing Wei
;
David W. Piotrowski
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 19:3328-3332
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7 .
Biochemical basis for differences in metabolism-dependent genotoxicity by two diazinylpiperazine-based 5-HT2C receptor agonists
저자
by
Jiri Aubrecht
;
Janvi Paralkar
;
Jonathan N. Bauman
;
Kim F. McClure
;
Santo R. Cortina
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 19:1559-1563
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