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1 .
Pharmacological inhibition of MERTK induces in vivo retinal degeneration: a multimodal imaging ocular safety assessment
저자
by
Gregory Hamm
;
Gareth Maglennon
;
Beth Williamson
;
Ruth Macdonald
;
Ann Doherty
, et al.
소스
Archives of Toxicology
. 96:613-624
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7 .
Optimization of an Imidazo[1,2-a]pyridine Series to Afford Highly Selective Type I1/2 Dual Mer/Axl Kinase Inhibitors with In Vivo Efficacy
저자
by
Edward J. Hennessy
;
Marianne Schimpl
;
Emma Rivers
;
Paul D. Smith
;
Elizabeth Hardaker
, et al.
소스
Journal of Medicinal Chemistry
. 64:13524-13539
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7 .
Identification and Strategies to Mitigate High Total Clearance of Benzylamine-Substituted Biphenyl Ring Systems
저자
by
Beth Williamson
;
Lindsay McMurray
;
Scott Boyd
;
Olga Collingwood
;
Neville McLean
, et al.
소스
Molecular pharmaceutics
. 19(7)
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7 .
A-loop interactions in Mer tyrosine kinase give rise to inhibitors with two-step mechanism and long residence time of binding
저자
by
William McCoull
;
Jon Winter-Holt
;
Marianne Schimpl
;
Elizabeth Underwood
;
Ross Overman
, et al.
소스
Biochemical Journal
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7 .
Discovery of (2R)-N-[3-[2-[(3-Methoxy-1-methyl-pyrazol-4-yl)amino]pyrimidin-4-yl]-1H-indol-7-yl]-2-(4-methylpiperazin-1-yl)propenamide (AZD4205) as a Potent and Selective Janus Kinase 1 Inhibitor
저자
by
Nanhua Deng
;
Sameer Kawatkar
;
Haoyu Wang
;
Michael Zinda
;
Allan Wu
, et al.
소스
Journal of Medicinal Chemistry
. 63:4517-4527
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7 .
Generating Selective Leads for Mer Kinase Inhibitors-Example of a Comprehensive Lead-Generation Strategy
저자
by
Ross Overman
;
Juli Warwicker
;
Kristin Goldberg
;
Alexander Pflug
;
Jeremy S. Disch
, et al.
소스
Journal of medicinal chemistry
. 64(6)
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7 .
A High-Throughput Screening Triage Workflow to Authenticate a Novel Series of PFKFB3 Inhibitors
저자
by
Ian M. Hardern
;
Jarrod Walsh
;
Ed Wheatley
;
Jon Winter-Holt
;
Sarita Maman
, et al.
소스
SLAS discovery : advancing life sciences RD
. 23(1)
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7 .
Abstract 979: Discovery of the JAK1 selective kinase inhibitor AZD4205
저자
by
Sameer Kawatkar
;
Kristen Bell
;
Richard Woessner
;
Neil P. Grimster
;
Qibin Su
, et al.
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Cancer Research
. 77:979-979
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7 .
MTH1 Substrate Recognition—An Example of Specific Promiscuity
저자
by
Jonathan Read
;
Jason Breed
;
J. Willem M. Nissink
;
Michal Bista
;
Jon Winter-Holt
, et al.
소스
PLoS ONE
PLoS ONE, Vol 11, Iss 3, p e0151154 (2016)
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