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1 . Academic Journal
Silencing Myostatin Using Cholesterol-conjugated siRNAs Induces Muscle Growth
저자
by
Tayeba Khan
;
Hans Weber
;
Jillian DiMuzio
;
Andrea Matter
;
Belma Dogdas
, et al.
소스
Molecular Therapy: Nucleic Acids, Vol 5, Iss C (2016)
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7 . Academic Journal
Proof-of-concept Studies for siRNA-mediated Gene Silencing for Coagulation Factors in Rat and Rabbit
저자
by
Zhu Chen
;
Bin Luo
;
Tian-Quan Cai
;
Anil Thankappan
;
Yiming Xu
, et al.
소스
Molecular Therapy: Nucleic Acids, Vol 4, Iss C (2015)
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7 .
823 IMM20059, a novel anti-EPN1 antibody, in combination with atezolizumab significantly enhances tumor regression in the B16.F10 syngeneic melanoma model compared to anti-PD-L1 monotherapy
저자
by
John Dowling
;
Pavel Nikitin
;
Cezary Swider
;
Chris Nicolescu
;
Halley Shukla
, et al.
소스
Regular and Young Investigator Award Abstracts
.
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7 .
Systematic chemical modifications of single stranded siRNAs significantly improved CTNNB1 mRNA silencing
저자
by
Laura Sepp-Lorenzino
;
Hangchun Zhang
;
Yi Pei
;
South Victoria J
;
Steven L. Colletti
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 26:4513-4517
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7 .
Identification and in Vivo Evaluation of Liver X Receptor β-Selective Agonists for the Potential Treatment of Alzheimer’s Disease
저자
by
Kausik K. Nanda
;
Yang Yuan
;
Celina Zerbinatti
;
Zhongguo Chen
;
Yingjie Li
, et al.
소스
Journal of Medicinal Chemistry
. 59:3489-3498
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7 .
P2-Quinazolinones and Bis-Macrocycles as New Templates for Next-Generation Hepatitis C Virus NS3/4a Protease Inhibitors: Discovery of MK-2748 and MK-6325
저자
by
Anne Taylor
;
Charles J. Mcintyre
;
Christine Fandozzi
;
Carolyn McHale
;
Jillian DiMuzio
, et al.
소스
ChemMedChem
. 10:727-735
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7 .
siRNA-Mediated Knockdown of P450 Oxidoreductase in Rats: A Tool to Reduce Metabolism by CYPs and Increase Exposure of High Clearance Compounds
저자
by
Brian A. Carr
;
Inthirai Somasuntharam
;
Traci Q. Lifsted
;
Martha A. DiPietro
;
Christopher R. Gibson
, et al.
소스
Pharmaceutical Research
. 31:3445-3460
Full Text (Springer)
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7 .
Development of macrocyclic inhibitors of HCV NS3/4A protease with cyclic constrained P2–P4 linkers
저자
by
John A. McCauley
;
Kevin Nguyen
;
Anne Taylor
;
Joseph J. Romano
;
Steven S. Carroll
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 22:7207-7213
Web of Science
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7 .
Silencing Myostatin Using Cholesterol-conjugated siRNAs Induces Muscle Growth
저자
by
Anil Thankappan
;
Laura Sepp-Lorenzino
;
Andrea Matter
;
Vasant Jadhav
;
Tosha Shah
, et al.
소스
Molecular Therapy. Nucleic Acids
Molecular Therapy: Nucleic Acids, Vol 5, Iss C (2016)
Full Text (ScienceDirect)
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7 .
Discovery of MK-1220: A Macrocyclic Inhibitor of Hepatitis C Virus NS3/4A Protease with Improved Preclinical Plasma Exposure
저자
by
John Swestock
;
Christine Fandozzi
;
John A. McCauley
;
Nicole Trainor
;
Bang-Lin Wan
, et al.
소스
ACS Medicinal Chemistry Letters
. 2:207-212
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