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1 .
Dual Inhibition of TYK2 and JAK1 for the Treatment of Autoimmune Diseases: Discovery of ((S)-2,2-Difluorocyclopropyl)((1R,5S)-3-(2-((1-methyl-1H-pyrazol-4-yl)amino)pyrimidin-4-yl)-3,8-diazabicyclo[3.2.1]octan-8-yl)methanone (PF-06700841)
저자
by
Brett D. Hollingshead
;
Fabien Vincent
;
Tsung H. Lin
;
John I. Trujillo
;
Betsy Pierce
, et al.
소스
Journal of Medicinal Chemistry
. 61:8597-8612
Web of Science
Scopus
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7 .
Discovery of a Potent and Selective Sphingosine Kinase 1 Inhibitor through the Molecular Combination of Chemotype-Distinct Screening Hits
저자
by
Maureen K. Highkin
;
Matthew D. McReynolds
;
Matthew J. Saabye
;
John W. Rains
;
Kaliapan Iyanar
, et al.
소스
Journal of medicinal chemistry
. 60(6)
Scopus
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7 .
Design of a Janus Kinase 3 (JAK3) Specific Inhibitor 1-((2S,5R)-5-((7H-Pyrrolo[2,3-d]pyrimidin-4-yl)amino)-2-methylpiperidin-1-yl)prop-2-en-1-one (PF-06651600) Allowing for the Interrogation of JAK3 Signaling in Humans
저자
by
Louis Leung
;
Jonathan Langille
;
John I. Trujillo
;
Paul B. Balbo
;
Jason Jussif
, et al.
소스
Journal of medicinal chemistry
. 60(5)
Scopus
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7 .
Design and Synthesis of a Pan-Janus Kinase Inhibitor Clinical Candidate (PF-06263276) Suitable for Inhaled and Topical Delivery for the Treatment of Inflammatory Diseases of the Lungs and Skin
저자
by
Iain Kilty
;
Yogesh A. Sabnis
;
Paul Morgan
;
Jill Chrencik
;
Florian Wakenhut
, et al.
소스
Journal of medicinal chemistry
. 60(2)
Open Access (OpenAIRE)
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7 .
Modulation of cellular S1P levels with a novel, potent and specific inhibitor of sphingosine kinase-1
저자
by
Michelle Kraus
;
Jay M. Wendling
;
Olga V. Nemirovskiy
;
John W. Rains
;
Vincent Peterkin
, et al.
소스
Biochemical Journal
. 444:79-88
Web of Science
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7 .
Structural and Thermodynamic Characterization of the TYK2 and JAK3 Kinase Domains in Complex with CP-690550 and CMP-6
저자
by
James R. Kiefer
;
Joseph W. Leone
;
Alfredo G. Tomasselli
;
Robin A. Weinberg
;
Akshay Patny
, et al.
소스
Journal of Molecular Biology
. 400:413-433
Web of Science
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7 .
Expression, purification, and characterization of TYK-2 kinase domain, a member of the Janus kinase family
저자
by
Thomas L. Emmons
;
Alfredo G. Tomasselli
;
Robin A. Weinberg
;
H. David Fischer
;
Jill Chrencik
, et al.
소스
Biochemical and Biophysical Research Communications
. 396:543-548
Web of Science
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7 .
Expression, purification, characterization and crystallization of non- and phosphorylated states of JAK2 and JAK3 kinase domain
저자
by
Thomas L. Emmons
;
James R. Kiefer
;
Joseph W. Leone
;
John F. Schindler
;
Melissa S. Harris
, et al.
소스
Protein Expression and Purification
. 69:54-63
Web of Science
Scopus
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7 .
Structure of human ADAM-8 catalytic domain complexed with batimastat
저자
by
James R. Kiefer
;
D.H. Fischer
;
Jennifer M. Williams
;
Huey-Sheng Shieh
;
Jill Chrencik
, et al.
소스
Acta crystallographica. Section F, Structural biology and crystallization communications
. 68(Pt 6)
Open Access (OpenAIRE)
Scopus
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7 .
Novel insights into the cellular mechanisms of the anti-inflammatory effects of NF-kappaB essential modulator binding domain peptides
저자
by
Sumathy Mathialagan
;
Jill Chrencik
;
Scott S. Woodard
;
Nandini Kishore
;
Julia A. Guzova
, et al.
소스
The Journal of Biological Chemistry
Full Text (ScienceDirect)
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