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1 . Academic Journal
Recent advances in the molecular design and applications of viral RNA-targeting antiviral modalities
저자
by
Dai, Jiaojiao
;
Jiang, Xiangyi
;
da Silva-Júnior, Edeildo Ferreira
;
Du, Shaoqing
;
Liu, Xinyong
, et al.
소스
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Drug Discovery Today
August 2024 29(8)
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7 . Academic Journal
Discovery of potent HIV-1 NNRTIs by CuAAC click-chemistry-based miniaturized synthesis, rapid screening and structure optimization
저자
by
Jing, Lanlan
;
Wu, Gaochan
;
Zhao, Fabao
;
Jiang, Xiangyi
;
Liu, Na
, et al.
소스
In
European Journal of Medicinal Chemistry
5 November 2024 277
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7 . Academic Journal
Discovery of novel diarypyrimidine derivatives bearing six-membered non-aromatic heterocycles as potent HIV-1 NNRTIs with improved anti-resistance and drug-like profiles
저자
by
Jiang, Xiangyi
;
Huang, Boshi
;
Zalloum, Waleed A.
;
Chen, Chin-Ho
;
Ji, Xiangkai
, et al.
소스
In
European Journal of Medicinal Chemistry
5 October 2023 258
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7 . Academic Journal
Design, synthesis, and biological evaluation of novel sulfamoylbenzamide derivatives as HBV capsid assembly modulators
저자
by
Wang, Shuo
;
Ren, Yujie
;
Li, Qilan
;
Wang, Ya
;
Jiang, Xiangyi
, et al.
소스
In
Bioorganic Chemistry
December 2022 129
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7 . Academic Journal
Design, synthesis, and mechanistic investigations of phenylalanine derivatives containing a benzothiazole moiety as HIV-1 capsid inhibitors with improved metabolic stability
저자
by
Xu, Shujing
;
Sun, Lin
;
Dick, Alexej
;
Zalloum, Waleed A.
;
Huang, Tianguang
, et al.
소스
In
European Journal of Medicinal Chemistry
5 January 2022 227
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7 . Academic Journal
Design, synthesis, and mechanism study of dimerized phenylalanine derivatives as novel HIV-1 capsid inhibitors
저자
by
Zhang, Xujie
;
Sun, Lin
;
Meuser, Megan E.
;
Zalloum, Waleed A.
;
Xu, Shujing
, et al.
소스
In
European Journal of Medicinal Chemistry
15 December 2021 226
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7 . Academic Journal
Exploiting the tolerant region I of the non-nucleoside reverse transcriptase inhibitor (NNRTI) binding pocket. Part 2: Discovery of diarylpyrimidine derivatives as potent HIV-1 NNRTIs with high Fsp3 values and favorable drug-like properties
저자
by
Jiang, Xiangyi
;
Huang, Boshi
;
Olotu, Fisayo A.
;
Li, Jing
;
Kang, Dongwei
, et al.
소스
In
European Journal of Medicinal Chemistry
5 March 2021 213
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7 . Academic Journal
Targeting dual tolerant regions of binding pocket: Discovery of novel morpholine-substituted diarylpyrimidines as potent HIV-1 NNRTIs with significantly improved water solubility
저자
by
Wang, Zhao
;
Kang, Dongwei
;
Feng, Da
;
Cherukupalli, Srinivasulu
;
Jiang, Xiangyi
, et al.
소스
In
European Journal of Medicinal Chemistry
15 November 2020 206
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7 . Academic Journal
In situ click chemistry-based rapid discovery of novel HIV-1 NNRTIs by exploiting the hydrophobic channel and tolerant regions of NNIBP
저자
by
Kang, Dongwei
;
Feng, Da
;
Jing, Lanlan
;
Sun, Yanying
;
Wei, Fenju
, et al.
소스
In
European Journal of Medicinal Chemistry
1 May 2020 193
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7 . Academic Journal
Discovery of novel “Dual-site” binding oseltamivir derivatives as potent influenza virus neuraminidase inhibitors
저자
by
Ai, Wei
;
Zhang, Jian
;
Zalloum, Waleed A.
;
Jia, Ruifang
;
Cherukupalli, Srinivasulu
, et al.
소스
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European Journal of Medicinal Chemistry
1 April 2020 191
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