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1 . Academic Journal
A GRM7 mutation associated with developmental delay reduces mGlu7 expression and produces neurological phenotypes
저자
by
Nicole M. Fisher
;
Aqeela AlHashim
;
Aditi B. Buch
;
Hana Badivuku
;
Manar M. Samman
, et al.
소스
JCI Insight, Vol 6, Iss 4 (2021)
Open Access (DOAJ)
Web of Science
Scopus
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7 .
Discovery of VU6028418: A Highly Selective and Orally Bioavailable M4 Muscarinic Acetylcholine Receptor Antagonist
저자
by
Sichen Chang
;
Jonathan W. Dickerson
;
Baker Logan A
;
Thomas M. Bridges
;
Craig W. Lindsley
, et al.
소스
ACS Med Chem Lett
Open Access (OpenAIRE)
Web of Science
Scopus
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7 .
Discovery of the First Selective M4 Muscarinic Acetylcholine Receptor Antagonists with in Vivo Antiparkinsonian and Antidystonic Efficacy
저자
by
Jerri M. Rook
;
Aaron M. Bender
;
Colleen M. Niswender
;
Yuping Donsante
;
P. Jeffrey Conn
, et al.
소스
ACS Pharmacology & Translational Science
. 4:1306-1321
Open Access (OpenAIRE)
Scopus
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7 .
Hyperactive Striatal Dopamine Signaling Observed in Huntington’s Disease Mouse Models Prior to Motor Symptom Onset Can be Attenuated via Activation of M 4 Receptors
저자
by
Roland M. Rodriguez
;
Daniel J. Foster
;
Madigan L. Lavery
;
Curran M. Johnston
;
Mark S. Moehle
, et al.
소스
The FASEB Journal
. 36
Scopus
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7 .
CB2 Receptor Potentiation Mediates Antipsychotic‐like Efficacy in Mice
저자
by
Anthony S. Ferranti
;
Tazeen Ishmam
;
Isaiah C. Swann
;
Jennifer Du
;
Janet Mariadoss
, et al.
소스
The FASEB Journal
. 36
Scopus
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7 . Academic Journal
Development ofNovel, CNS Penetrant Positive AllostericModulators for the Metabotropic Glutamate Receptor Subtype 1 (mGlu1), Based on an N-(3-Chloro-4-(1,3-dioxoisoindolin-2-yl)phenyl)-3-methylfuran-2-carboxamideScaffold, That Potentiate Wild Type and Mutant mGlu1ReceptorsFound in Schizophrenics
저자
by
PedroM. Garcia-Barrantes
;
Hyekyung P. Cho
;
Colleen M. Niswender
;
FrankW. Byers
;
Charles W. Locuson
, et al.
소스
Journal of Medicinal Chemistry
. Oct2015, Vol. 58 Issue 20, p7959-7971. 13p.
Full Text (ACS)
Web of Science
Scopus
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7 .
A GRM7 mutation associated with developmental delay reduces mGlu7 expression and produces neurological phenotypes
저자
by
Mark D. Does
;
Jerri M. Rook
;
Aditi B. Buch
;
Kelly M. Weiss
;
Manar M. Samman
, et al.
소스
JCI Insight, Vol 6, Iss 4 (2021)
JCI Insight
Open Access (OpenAIRE)
Scopus
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7 .
VU6007477, a Novel M1 PAM Based on a Pyrrolo[2,3-b]pyridine Carboxamide Core Devoid of Cholinergic Adverse Events
저자
by
Anna L. Blobaum
;
Jerri M. Rook
;
Jonathan W. Dickerson
;
Colleen M. Niswender
;
Julie L. Engers
, et al.
소스
ACS Medicinal Chemistry Letters
. 9:917-922
Open Access (OpenAIRE)
Web of Science
Scopus
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7 .
Safety and pharmacokinetics of the muscarinic positive allosteric modulator VU319: A phase 1 single dose study
저자
by
Jerri M. Rook
;
Alexandra P. Key
;
Alexander C. Conley
;
Jennifer Urbano Blackford
;
Craig W. Lindsley
, et al.
소스
Alzheimer's & Dementia
. 16
Open Access (OpenAIRE)
Scopus
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7 .
Cognitive performance effects following a single dose of the M 1 muscarinic positive allosteric modulator VU319
저자
by
Jerri M. Rook
;
Craig W. Lindsley
;
Paul A. Newhouse
;
Carrie K. Jones
;
Alexandra P. Key
, et al.
소스
Alzheimer's & Dementia
. 16
Open Access (OpenAIRE)
Scopus
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