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1 . Academic Journal
Fc-GDF15 glyco-engineering and receptor binding affinity optimization for body weight regulation
저자
by
Ella Fung
;
Liya Kang
;
Diana Sapashnik
;
Susan Benard
;
Annette Sievers
, et al.
소스
Scientific Reports, Vol 11, Iss 1, Pp 1-12 (2021)
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7 . Academic Journal
A Mechanistic Site-Of-Action Model: A Tool for Informing Right Target, Right Compound, And Right Dose for Therapeutic Antagonistic Antibody Programs
저자
by
Georgi I. Kapitanov
;
Jeffrey R. Chabot
;
Jatin Narula
;
Mahua Roy
;
Hendrik Neubert
, et al.
소스
Frontiers in Bioinformatics, Vol 1 (2021)
Open Access (DOAJ)
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7 .
A Mechanistic Site-Of-Action Model: A Tool for Informing Right Target, Right Compound, And Right Dose for Therapeutic Antagonistic Antibody Programs
저자
by
Hannah M. Jones
;
Hendrik Neubert
;
Mahua Roy
;
Vahid Farrokhi
;
Jatin Narula
, et al.
소스
Frontiers in Bioinformatics, Vol 1 (2021)
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7 .
Small Molecule Proprotein Convertase Subtilisin/Kexin Type 9 (PCSK9) Inhibitors: Hit to Lead Optimization of Systemic Agents
저자
by
Liuqing Wei
;
Jun Xiao
;
Joseph S. Warmus
;
Jeffrey R. Chabot
;
Robert Dullea
, et al.
소스
Journal of Medicinal Chemistry
. 61:5704-5718
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7 .
Assessing the Feasibility of Neutralizing Osteopontin with Various Therapeutic Antibody Modalities
저자
by
Jeffrey R. Chabot
;
Vahid Farrokhi
;
Zhiyong Yang
;
Hendrik Neubert
.
소스
Scientific Reports, Vol 8, Iss 1, Pp 1-7 (2018)
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6 .
Liver-Targeted Small-Molecule Inhibitors of Proprotein Convertase Subtilisin/Kexin Type 9 Synthesis
저자
by
Dennis O. Scott
;
Spiros Liras
;
Roger B. Ruggeri
;
Heather Eng
;
Adam S. Kamlet
, et al.
소스
Angewandte Chemie International Edition
. 56:16218-16222
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7 . Academic Journal
Analysis of Mechanistic Pathway Models in Drug Discovery: p38 Pathway.
저자
by
Bart S. Hendriks
;
Fei Hua
;
Jeffrey R. Chabot
.
소스
Biotechnology Progress; Feb2008, Vol. 24 Issue 1, p96-109, 14p
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5 .
Once‐weekly administration of a long‐acting fibroblast growth factor 21 analogue modulates lipids, bone turnover markers, blood pressure and body weight differently in obese people with hypertriglyceridaemia and in non‐human primates
저자
by
Saswata Talukdar
;
Yan Weng
;
Jennifer Q. Dong
;
Veena Somayaji
;
Timothy P. Rolph
, et al.
소스
Diabetes, Obesity and Metabolism
. 19:1762-1772
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7 .
Examination of the Human Cytochrome P4503A4 Induction Potential of PF-06282999, an Irreversible Myeloperoxidase Inactivator: Integration of Preclinical, In Silico, and Biomarker Methodologies in the Prediction of the Clinical Outcome
저자
by
James R. Gosset
;
Zhiwu Lin
;
Jeffrey R. Chabot
;
Odette A. Fahmi
;
Albert M. Kim
, et al.
소스
Drug Metabolism and Disposition
. 45:501-511
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7 .
Physiologically relevant binding affinity quantification of monoclonal antibody PF-00547659 to mucosal addressin cell adhesion molecule forin vitro in vivocorrelation
저자
by
Christopher Lepsy
;
Jeffrey R. Chabot
;
Mireia Fernández Ocaña
;
Denise O'Hara
;
Darryl J. Bornhop
, et al.
소스
British Journal of Pharmacology
. 174:70-81
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