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1 .
Discovery and characterization of a selective IKZF2 glue degrader for cancer immunotherapy
저자
by
Simone Bonazzi
;
Eva d’Hennezel
;
Rohan E.J. Beckwith
;
Lei Xu
;
Aleem Fazal
, et al.
소스
Cell Chemical Biology
. 30:235-247.e12
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7 .
Targeted degradation of IKZF2 for cancer immunotherapy
저자
by
Jonathan Solomon
;
Simone Bonazzi
;
Eva d'Hennezel
;
Rohan Beckwith
;
Lei Xu
, et al.
소스
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7 .
Palladium Catalyzed C−O Coupling of Amino Alcohols for the Synthesis of Aryl Ethers
저자
by
Sanchez Carina Cristina
;
Jay Larrow
;
Cary Fridrich
;
Malte S. Mikus
.
소스
Advanced Synthesis & Catalysis
. 362:430-436
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6 .
Identification of TNO155, an Allosteric SHP2 Inhibitor for the Treatment of Cancer
저자
by
Kelly Slocum
;
Jianmei Fan
;
Michael Dore
;
Palermo Mark G
;
Zhan Deng
, et al.
소스
Journal of medicinal chemistry
. 63(22)
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7 .
Allosteric Inhibition of SHP2: Identification of a Potent, Selective, and Orally Efficacious Phosphatase Inhibitor
저자
by
Matthew J. LaMarche
;
Peter Fekkes
;
Jorge Garcia Fortanet
;
Michael Shultz
;
Denise Grunenfelder
, et al.
소스
Journal of Medicinal Chemistry
. 59:7773-7782
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7 .
Allosteric inhibition of SHP2 phosphatase inhibits cancers driven by receptor tyrosine kinases
저자
by
Palermo Mark G
;
Timothy Michael Ramsey
;
Ping Zhu
;
Shumei Liu
;
Jay Larrow
, et al.
소스
Nature
. 535:148-152
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7 .
COUNTERION QUANTIFICATION FOR DISCOVERY CHEMISTRY AND PRE-FORMULATION SALT SCREENING
저자
by
Lipa Shah
;
Thierry Mann
;
Penny Wright
;
Jennifer Bilotta
;
Joseph Twomey
, et al.
소스
Journal of Liquid Chromatography & Related Technologies
. 35:1001-1010
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7 .
Comparison of Large-Scale Routes to Manufacture Chiral exo-2-Norbornyl Thiourea
저자
by
James K. Lee
;
Pilar Franco
;
Geoffrey B. Cox
;
Kenichi Sakai
;
Jay Larrow
, et al.
소스
Organic Process Research & Development
. 14:133-141
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7 .
Discovery and Optimization of Triazolopyridazines as Potent and Selective Inhibitors of the c-Met Kinase
저자
by
Steven F. Bellon
;
Monica Reese
;
Jay Larrow
;
Isabelle Dussault
;
Stephanie Springer
, et al.
소스
Journal of Medicinal Chemistry
. 51:2879-2882
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7 .
Novel 2,3-Dihydro-1,4-Benzoxazines as Potent and Orally Bioavailable Inhibitors of Tumor-Driven Angiogenesis
저자
by
Shaun Flynn
;
James Bready
;
Shawn Harriman
;
Vinod F. Patel
;
Zhiyang Zhao
, et al.
소스
Journal of Medicinal Chemistry
. 51:1695-1705
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