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1 . Academic Journal
Tryptophan Substitution in CJ-15,208 (cyclo[Phe-D-Pro-Phe-Trp]) Introduces δ-Opioid Receptor Antagonism, Preventing Antinociceptive Tolerance and Stress-Induced Reinstatement of Extinguished Cocaine-Conditioned Place Preference
저자
by
Kristen H. Scherrer
;
Shainnel O. Eans
;
Jessica M. Medina
;
Sanjeewa N. Senadheera
;
Tanvir Khaliq
, et al.
소스
Pharmaceuticals, Vol 16, Iss 9, p 1218 (2023)
Open Access (DOAJ)
Web of Science
Scopus
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7 . Academic Journal
Quantification of kappa opioid receptor ligand potency, efficacy and desensitization using a real-time membrane potential assay
저자
by
Yuanzi Zhao
;
Anand A. Joshi
;
Jane V. Aldrich
;
Thomas F. Murray
.
소스
Biomedicine & Pharmacotherapy, Vol 143, Iss , Pp 112173- (2021)
Full Text (ScienceDirect)
Full Text (Clinical Key)
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Full Text (ScienceDirect O/A)
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6 . Academic Journal
Phenylalanine Stereoisomers of CJ-15,208 and [d-Trp]CJ-15,208 Exhibit Distinctly Different Opioid Activity Profiles
저자
by
Ariana C. Brice-Tutt
;
Sanjeewa N. Senadheera
;
Michelle L. Ganno
;
Shainnel O. Eans
;
Tanvir Khaliq
, et al.
소스
Molecules, Vol 25, Iss 17, p 3999 (2020)
Open Access (DOAJ)
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7 .
Analogs of the κ opioid receptor antagonist arodyn cyclized by ring-closing metathesis retain κ opioid receptor affinity, selectivity and κ opioid receptor antagonism
저자
by
Wei Jie Fang
;
Jane V. Aldrich
;
Thomas F. Murray
.
소스
Medicinal Chemistry Research
. 30:1397-1407
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5 .
Conformational Constraint between Aromatic Residue Side Chains in the 'Message' Sequence of the Peptide Arodyn Using Ring Closing Metathesis Results in a Potent and Selective Kappa Opioid Receptor Antagonist
저자
by
Jane V. Aldrich
;
Solomon A. Gisemba
;
Thomas F. Murray
;
Michael J. Ferracane
.
소스
Journal of Medicinal Chemistry
. 64:3153-3164
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6 .
An analog of [d-Trp]CJ-15,208 exhibits kappa opioid receptor antagonism following oral administration and prevents stress-induced reinstatement of extinguished morphine conditioned place preference
저자
by
Ariana C. Brice-Tutt
;
Shainnel O. Eans
;
Dmitry Yakovlev
;
Jane V. Aldrich
;
Jay P. McLaughlin
.
소스
Pharmacology, biochemistry, and behavior
. 217
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7 .
Design, Synthesis, and Characterization of the Macrocyclic Tetrapeptide cyclo[Pro-Sar-Phe-
d
-Phe]: A Mixed Opioid Receptor Agonist–Antagonist Following Oral Administration
저자
by
Thomas F. Murray
;
Jeremy S. Coleman
;
Lisa L. Wilson
;
Jay P. McLaughlin
;
Shainnel O. Eans
, et al.
소스
ACS Chemical Neuroscience
. 11:1324-1336
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7 . Academic Journal
Structure–ActivityRelationships of the PeptideKappa Opioid Receptor Antagonist Zyklophin.
저자
by
AnandA. Joshi
;
Thomas F. Murray
;
Jane V. Aldrich
.
소스
Journal of Medicinal Chemistry
. Nov2015, Vol. 58 Issue 22, p8783-8795. 13p.
Full Text (ACS)
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5 .
Peptide Kappa Opioid Receptor Ligands and Their Potential for Drug Development
저자
by
Jane V. Aldrich
;
Jay P. McLaughlin
.
소스
The Kappa Opioid Receptor ISBN: 9783030890735
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4 .
Phenylalanine Stereoisomers of CJ-15,208 and [d-Trp]CJ-15,208 Exhibit Distinctly Different Opioid Activity Profiles
저자
by
Thomas F. Murray
;
Jay P. McLaughlin
;
Sanjeewa N. Senadheera
;
Shainnel O. Eans
;
Ariana C. Brice-Tutt
, et al.
소스
Molecules
Volume 25
Issue 17
Molecules, Vol 25, Iss 3999, p 3999 (2020)
Open Access (OpenAIRE)
Web of Science
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