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1 .
Discovery of RMC-5552, a Selective Bi-Steric Inhibitor of mTORC1, for the Treatment of mTORC1-Activated Tumors
저자
by
G. Leslie Burnett
;
Yu C. Yang
;
James B. Aggen
;
Jennifer Pitzen
;
Micah K. Gliedt
, et al.
소스
Journal of Medicinal Chemistry
. 66:149-169
Open Access (OpenAIRE)
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7 .
Optimization of LpxC Inhibitors for Antibacterial Activity and Cardiovascular Safety
저자
by
Frederick Cohen
;
James B. Aggen
;
Logan D. Andrews
;
Zahra Assar
;
Jen Boggs
, et al.
소스
ChemMedChem
. 14:1560-1572
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7 .
Author Correction: Selective inhibitors of mTORC1 activate 4EBP1 and suppress tumor growth
저자
by
Bianca J. Lee
;
Jacob A. Boyer
;
G. Leslie Burnett
;
Arun P. Thottumkara
;
Nidhi Tibrewal
, et al.
소스
Nature Chemical Biology
. 17:1209-1209
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7 .
Compound design guidelines for evading the efflux and permeation barriers of Escherichia coli with the oxazolidinone class of antibacterials: Test case for a general approach to improving whole cell Gram-negative activity
저자
by
Paola C. Zucchi
;
James B. Aggen
;
Bilyana N. Koleva
;
Andrew Spaulding
;
Harold D. Cooper
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 27:5310-5321
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7 .
Synthesis and Microbiological Evaluation of Novel Tetracyclic Fluoroquinolones
저자
by
Allan Scott Wagman
;
Sara Lopez
;
Lloyd J. Simons
;
James B. Aggen
;
Ryan Cirz
, et al.
소스
ChemMedChem
. 12:1687-1692
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7 .
Author Correction: Selective inhibitors of mTORC1 activate 4EBP1 and suppress tumor growth
저자
by
Jacqueline Smith
;
Nidhi Tibrewal
;
Adrian Liam Gill
;
Gert Kiss
;
Abby Marquez
, et al.
소스
Nature Chemical Biology
. 17:925-925
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7 .
Abstract PR04: 4EBP1 reactivation by potent and selective bi-steric inhibitors of mTORC1
저자
by
G. Leslie Burnett
;
Mark A. Goldsmith
;
Daphne Hsieh
;
Pete Wildes
;
Jacqueline Smith
, et al.
소스
Molecular Cancer Research
. 18:PR04-PR04
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7 .
Abstract IA17: Strategies to target the mTORC1/eIF4F axis in B-cell leukemia and lymphoma
저자
by
Jacqueline Smith
;
Amos Fung
;
Bianca J. Lee
;
Ze'ev Ronai
;
Honyin Chiu
, et al.
소스
Molecular Cancer Research
. 18:IA17-IA17
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7 .
Progress against Escherichia coli with the Oxazolidinone Class of Antibacterials: Test Case for a General Approach To Improving Whole-Cell Gram-Negative Activity
저자
by
James B. Aggen
;
Harold D. Cooper
;
Elizabeth B. Hirsch
;
Bilyana N. Koleva
;
Paola C. Zucchi
, et al.
소스
ACS Infectious Diseases
. 2:405-426
Web of Science
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7 .
Abstract B108: 4EBP3 mRNA as a biomarker of therapeutic response to treatment with mTORC1 inhibitors
저자
by
Bianca J. Lee
;
Ed Lorenzana
;
Mallika Singh
;
Robert J. Nichols
;
Jaqueline A.M. Smith
, et al.
소스
Molecular Cancer Therapeutics
. 18:B108-B108
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