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1 . Academic Journal
Inhibiting a dynamic viral protease by targeting a non-catalytic cysteine
저자
by
Hulce, Kaitlin R.
;
Jaishankar, Priyadarshini
;
Lee, Gregory M.
;
Bohn, Markus-Frederik
;
Connelly, Emily J.
, et al.
소스
In
Cell Chemical Biology
19 May 2022 29(5):785-798
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7 . Academic Journal
Activation of Caspase-6 Is Promoted by a Mutant Huntingtin Fragment and Blocked by an Allosteric Inhibitor Compound
저자
by
Ehrnhoefer, Dagmar E.
;
Skotte, Niels H.
;
Reinshagen, Jeanette
;
Qiu, Xiaofan
;
Windshügel, Björn
, et al.
소스
In
Cell Chemical Biology
19 September 2019 26(9):1295-1305
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7 . Academic Journal
Structure-Based Optimization of Covalent, Small-Molecule Stabilizers of the 14-3-3σ/ERα Protein–Protein Interaction from Nonselective Fragments.
저자
by
Konstantinidou, Markella
;
Visser, Emira J.
;
Vandenboorn, Edmee
;
Chen, Sheng
;
Jaishankar, Priyadarshini
, et al.
소스
Journal of the American Chemical Society; 9/20/2023, Vol. 145 Issue 37, p20328-20343, 16p
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7 . Academic Journal
From Tethered to Freestanding Stabilizers of 14‐3‐3 Protein‐Protein Interactions through Fragment Linking.
저자
by
Visser, Emira J.
;
Jaishankar, Priyadarshini
;
Sijbesma, Eline
;
Pennings, Marloes A. M.
;
Vandenboorn, Edmee M. F.
, et al.
소스
Angewandte Chemie
. 9/11/2023, Vol. 135 Issue 37, p1-9. 9p.
Full Text (Wiley)
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7 . Academic Journal
Engaging a Non-catalytic Cysteine Residue Drives Potent and Selective Inhibition of Caspase‑6.
저자
by
Van Horn, Kurt S.
;
Wang, Dongju
;
Medina-Cleghorn, Daniel
;
Lee, Peter S.
;
Bryant, Clifford
, et al.
소스
Journal of the American Chemical Society; 5/10/2023, Vol. 145 Issue 18, p10015-10021, 7p
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7 . Academic Journal
Heteroaryl Phosphonates as Noncovalent Inhibitors of Both Serine- and Metallocarbapenemases.
저자
by
Pemberton, Orville A.
;
Jaishankar, Priyadarshini
;
Akhtar, Afroza
;
Adams, Jessie L.
;
Shaw, Lindsey N.
, et al.
소스
Journal of Medicinal Chemistry; 9/26/2019, Vol. 62 Issue 18, p8480-8496, 17p
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7 . Academic Journal
Novel non-peptidic vinylsulfones targeting the S2 and S3 subsites of parasite cysteine proteases
저자
by
Bryant, Clifford
;
Kerr, Iain D.
;
Debnath, Moumita
;
Ang, Kenny K.H.
;
Ratnam, Joseline
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2009 19(21):6218-6221
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7 . Periodical
Cyanopyrrolidine Inhibitors of Ubiquitin Specific Protease 7 Mediate Desulfhydration of the Active-Site Cysteine
저자
by
Bashore, Charlene
;
Jaishankar, Priyadarshini
;
Skelton, Nicholas J.
;
Fuhrmann, Jakob
;
Hearn, Brian R.
, et al.
소스
ACS Chemical Biology; June 2020, Vol. 15 Issue: 6 p1392-1400, 9p
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7 . Academic Journal
Active-Site Druggability of Carbapenemases and Broad-Spectrum Inhibitor Discovery.
저자
by
Torelli, Nicholas J.
;
Akhtar, Afroza
;
DeFrees, Kyle
;
Jaishankar, Priyadarshini
;
Pemberton, Orville A.
, et al.
소스
ACS Infectious Diseases; 6/14/2019, Vol. 5 Issue 6, p1013-1, 9p
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7 . Academic Journal
Potency and selectivity of P2/P3-modified inhibitors of cysteine proteases from trypanosomes
저자
by
Jaishankar, Priyadarshini
;
Hansell, Elizabeth
;
Zhao, Dong-Mei
;
Doyle, Patricia S.
;
McKerrow, James H.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2008 18(2):624-628
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