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1 . Academic Journal
Site-directed deuteration of dronedarone preserves cytochrome P4502J2 activity and mitigates its cardiac adverse effects in canine arrhythmic hearts
저자
by
Aneesh V. Karkhanis
;
Gopalakrishnan Venkatesan
;
Ryuichi Kambayashi
;
Jacqueline Wen Hui Leow
;
Marcus Qingrui Han
, et al.
소스
Acta Pharmaceutica Sinica B, Vol 12, Iss 10, Pp 3905-3923 (2022)
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7 .
Development and verification of a physiologically based pharmacokinetic model of dronedarone and its active metabolite N‐desbutyldronedarone: Application to prospective simulation of complex drug–drug interaction with rivaroxaban
저자
by
Jacqueline Wen Hui Leow
;
Xiao Jun Ang
;
Eric Chun Yong Chan
.
소스
British Journal of Clinical Pharmacology
. 89:1873-1890
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5 .
Investigating the relevance of CYP2J2 inhibition for drugs known to cause intermediate to high risk torsades de pointes
저자
by
Jacqueline Wen Hui Leow
;
Yuxiang Gu
;
Eric Chun Yong Chan
.
소스
European Journal of Pharmaceutical Sciences
. 187:106475
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5 .
Atypical kinetics of cytochrome P450 enzymes in pharmacology and toxicology
저자
by
Jacqueline Wen Hui Leow
;
Lloyd Wei Tat Tang
;
Eric Chun Yong Chan
.
소스
Pharmacology and Toxicology of Cytochrome P450 – 60th Anniversary ISBN: 9780323911092
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5 .
Site-directed deuteration of dronedarone preserves cytochrome P4502J2 activity and mitigates its cardiac adverse effects in canine arrhythmic hearts
저자
by
Aneesh V. Karkhanis
;
Gopalakrishnan Venkatesan
;
Ryuichi Kambayashi
;
Jacqueline Wen Hui Leow
;
Marcus Qingrui Han
, et al.
소스
Acta pharmaceutica Sinica. B
. 12(10)
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7 .
How the Deuteration of Dronedarone Can Modify Its Cardiovascular Profile: In Vivo Characterization of Electropharmacological Effects of Poyendarone, a Deuterated Analogue of Dronedarone
저자
by
Koki Chiba
;
Eric Chun Yong Chan
;
Akio Matsumoto
;
Yoshio Nunoi
;
Mihoko Hagiwara-Nagasawa
, et al.
소스
Cardiovascular toxicology
. 20(4)
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7 .
Atypical Michaelis-Menten kinetics in cytochrome P450 enzymes: A focus on substrate inhibition
저자
by
Jacqueline Wen Hui Leow
;
Eric Chun Yong Chan
.
소스
Biochemical pharmacology
. 169
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4 .
Dronedarone-Induced Cardiac Mitochondrial Dysfunction and Its Mitigation by Epoxyeicosatrienoic Acids
저자
by
Eric Chun Yong Chan
;
Jacqueline Wen Hui Leow
;
Aneesh V. Karkhanis
;
Thilo Hagen
.
소스
Toxicological Sciences
. 163:79-91
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6 .
Atypical kinetics of cytochrome P450 2J2: Epoxidation of arachidonic acid and reversible inhibition by xenobiotic inhibitors
저자
by
Ravi Kumar Verma
;
Amos Boon Hao Lim
;
Hao Fan
;
Jacqueline Wen Hui Leow
;
Eric Chun Yong Chan
.
소스
European Journal of Pharmaceutical Sciences
. 164:105889
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7 .
P102 - Predicting risk of cardiac arrhythmias based on inhibitory potencies (Ki) against CYP2J2-mediated arachidonic acid metabolism
저자
by
Jacqueline Wen Hui Leow
;
Hao Fan
;
Ravi Kumar Verma
;
Eric Chun Yong Chan
;
Amos Boon Hao Lim
.
소스
Drug Metabolism and Pharmacokinetics
. 35:S53
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