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1 . Academic Journal
Discovery and mechanistic study of thiazole-4-acylsulfonamide derivatives as potent and orally active ChemR23 inhibitors with a long-acting effect in cynomolgus monkeys
저자
by
Imaizumi, Takamichi
;
Otsubo, Shigeki
;
Maemoto, Michihiro
;
Kobayashi, Atsuko
;
Komai, Masato
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 February 2022 56
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7 . Academic Journal
Corrigendum to “Discovery and mechanistic study of thiazole-4-acylsulfonamide derivatives as potent and orally active ChemR23 inhibitors with a long-acting effect in cynomolgus monkeys” [Bioorg. Med. Chem. 56 (2022) 116587]
저자
by
Imaizumi, Takamichi
;
Otsubo, Shigeki
;
Maemoto, Michihiro
;
Kobayashi, Atsuko
;
Komai, Masato
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 April 2022 59
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7 . Academic Journal
Irciniastatin A induces JNK activation that is involved in caspase-8-dependent apoptosis via the mitochondrial pathway
저자
by
Chinen, Takumi
;
Nagumo, Yoko
;
Watanabe, Tsubasa
;
Imaizumi, Takamichi
;
Shibuya, Masatoshi
, et al.
소스
In
Toxicology Letters
2010 199(3):341-346
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7 . Academic Journal
The synthesis and evaluation of the antiproliferative activity of deacidified GEX1A analogues.
저자
by
Imaizumi, Takamichi
;
Nakagawa, Hiroshi
;
Hori, Ran
;
Watanabe, Yasuo
;
Soga, Shiro
, et al.
소스
Journal of Antibiotics; May2017, Vol. 70 Issue 5, p675-679, 5p
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7 . Academic Journal
The design, synthesis and evaluation of 2-aminobenzoxazole analogues as potent and orally efficacious ChemR23 inhibitors
저자
by
Imaizumi, Takamichi
;
Otsubo, Shigeki
;
Komai, Masato
;
Takada, Hidenori
;
Maemoto, Michihiro
, et al.
소스
BIOORGANIC & MEDICINAL CHEMISTRY
; SEP 1 2020, 28 17, p115622 18p.
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7 . Academic Journal
Eu(OTf)3-Catalyzed Highly Regioselective Nucleophilic Ring Opening of 2,3-Epoxy Alcohols: An Efficient Entry to 3-Substituted 1,2-Diol Derivatives.
저자
by
Uesugi, Shun-ichiro
;
Watanabe, Tsubasa
;
Imaizumi, Takamichi
;
Shibuya, Masatoshi
;
Kanoh, Naoki
, et al.
소스
Organic Letters
. Sep2014, Vol. 16 Issue 17, p4408-4411. 4p.
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7 . Academic Journal
Nicotinamide phosphoribosyltransferase is a molecular target of potent anticancer agents identified from phenotype-based drug screening
저자
by
Yamaguchi, Daisuke
;
Imaizumi, Takamichi
;
Yagi, Kaori
;
Matsumoto, Yuichi
;
Nakashima, Takayuki
, et al.
소스
Scientific Reports
. 9(1)
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7 . Academic Journal
Syntheses and Biological Evaluation of Irciniastatin A and the C1−C2 Alkyne Analogue.
저자
by
Watanabe, Tsubasa
;
Imaizumi, Takamichi
;
Chinen, Takumi
;
Nagumo, Yoko
;
Shibuya, Masatoshi
, et al.
소스
Organic Letters
. Mar2010, Vol. 12 Issue 5, p1040-1043. 4p.
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7 . Academic Journal
The discovery and optimization of a series of 2-aminobenzoxazole derivatives as ChemR23 inhibitors.
저자
by
Imaizumi, Takamichi
;
Kobayashi, Atsuko
;
Otsubo, Shigeki
;
Komai, Masato
;
Magara, Megumiko
, et al.
소스
Bioorganic & Medicinal Chemistry
. Nov2019, Vol. 27 Issue 21, pN.PAG-N.PAG. 1p.
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7 . Academic Journal
Total Synthesis and Biological Evaluation of Irciniastatin A (a.k.a. Psymberin) and Irciniastatin B
저자
by
Uesugi, Shun-ichiro
;
Watanabe, Tsubasa
;
Imaizumi, Takamichi
;
Ota, Yu
;
Yoshida, Keisuke
, et al.
소스
JOURNAL OF ORGANIC CHEMISTRY
; DEC 18 2015, 80 24, p12333-p12350, 18p.
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