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1 . Academic Journal
Phosphoinositide-3-kinase inhibitors: Evaluation of substituted alcohols as replacements for the piperazine sulfonamide portion of AMG 511
저자
by
Lanman, Brian A.
;
Reed, Anthony B.
;
Cee, Victor J.
;
Hong, Fang-Tsao
;
Pettus, Liping H.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 December 2014 24(24):5630-5634
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7 . Academic Journal
Discovery of Selective Pituitary Adenylate Cyclase 1 Receptor (PAC1R) Antagonist Peptides Potent in a Maxadilan/PACAP38-Induced Increase in Blood Flow Pharmacodynamic Model.
저자
by
Hu, Essa
;
Hong, Fang-Tsao
;
Aral, Jennifer
;
Long, Jason
;
Piper, Derek E.
, et al.
소스
Journal of Medicinal Chemistry; 3/25/2021, Vol. 64 Issue 6, p3427-3438, 12p
Full Text (ACS)
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7 . Academic Journal
Azole-based inhibitors of AKT/PKB for the treatment of cancer
저자
by
Zeng, Qingping
;
Allen, John G.
;
Bourbeau, Matthew P.
;
Wang, Xianghong
;
Yao, Guomin
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
2010 20(5):1559-1564
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7 . Academic Journal
Small Molecule Disruptors of the Glucokinase–GlucokinaseRegulatory Protein Interaction: 4. Exploration of a Novel BindingPocket.
저자
by
Hong, Fang-Tsao
;
Norman, Mark H.
;
Ashton, Kate S.
;
Bartberger, Michael D.
;
Chen, Jie
, et al.
소스
Journal of Medicinal Chemistry
. Jul2014, Vol. 57 Issue 14, p5949-5964. 16p.
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7 . Academic Journal
Small Molecule Disruptorsof the Glucokinase–GlucokinaseRegulatory Protein Interaction: 2. Leveraging Structure-Based DrugDesign to Identify Analogues with Improved Pharmacokinetic Profiles.
저자
by
St. Jean, David J.
;
Ashton, Kate S.
;
Bartberger, Michael D.
;
Chen, Jie
;
Chmait, Samer
, et al.
소스
Journal of Medicinal Chemistry
. Jan2014, Vol. 57 Issue 2, p325-338. 14p.
Full Text (ACS)
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7 . Academic Journal
Selective Class I Phosphoinositide3-KinaseInhibitors: Optimization of a Series of Pyridyltriazines Leading tothe Identification of a Clinical Candidate, AMG 511.
저자
by
Norman, Mark H.
;
Andrews, Kristin L.
;
Bo, Yunxin Y.
;
Booker, Shon K.
;
Caenepeel, Sean
, et al.
소스
Journal of Medicinal Chemistry
. Sep2012, Vol. 55 Issue 17, p7796-7816. 21p.
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7 . Academic Journal
Structure-Based Designof a Novel Series of Potent, Selective Inhibitors of the Class IPhosphatidylinositol 3-Kinases.
저자
by
Smith, Adrian L.
;
DâAngelo, Noel D.
;
Bo, Yunxin Y.
;
Booker, Shon K.
;
Cee, Victor J.
, et al.
소스
Journal of Medicinal Chemistry
. Jun2012, Vol. 55 Issue 11, p5188-5219. 32p.
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7 . Academic Journal
Discovery and Structure-Guided Optimization of Diarylmethanesulfonamide Disrupters of Glucokinase-Glucokinase Regulatory Protein (GK-GKRP) Binding: Strategic Use of a N -> S (n(N) -> sigma*(S-X)) Interaction for Conformational Constraint
저자
by
Pennington, Lewis D.
;
Bartberger, Michael D.
;
Croghan, Michael D.
;
Andrews, Kristin L.
;
Ashton, Kate S.
, et al.
소스
JOURNAL OF MEDICINAL CHEMISTRY
; DEC 24 2015, 58 24, p9663-p9679, 17p.
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7 . Academic Journal
Oxopyrido[2,3-d]pyrimidines as Covalent L858R/T790M Mutant Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors
저자
by
Wurz, Ryan P.
;
Pettus, Liping H.
;
Ashton, Kate
;
Brown, James
;
Chen, Jian Jeffrey
, et al.
소스
ACS MEDICINAL CHEMISTRY LETTERS
; SEP 2015, 6 9, p987-p992, 6p.
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7 . Academic Journal
Small Molecule Disruptors of the Glucokinase-Glucokinase Regulatory Protein Interaction: 5. A Novel Aryl Sulfone Series, Optimization Through Conformational Analysis
저자
by
Tamayo, Nuria A.
;
Norman, Mark H.
;
Bartberger, Michael D.
;
Hong, Fang-Tsao
;
Bo, Yunxin
, et al.
소스
JOURNAL OF MEDICINAL CHEMISTRY
; JUN 11 2015, 58 11, p4462-p4482, 21p.
Full Text (ACS)
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