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1 . Academic Journal
Structural basis of ligand recognition and design of antihistamines targeting histamine H4 receptor
저자
by
Ruixue Xia
;
Shuang Shi
;
Zhenmei Xu
;
Henry F. Vischer
;
Albert D. Windhorst
, et al.
소스
Nature Communications, Vol 15, Iss 1, Pp 1-13 (2024)
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7 . Academic Journal
Multiplex Detection of Fluorescent Chemokine Binding to CXC Chemokine Receptors by NanoBRET
저자
by
Justyna M. Adamska
;
Spyridon Leftheriotis
;
Reggie Bosma
;
Henry F. Vischer
;
Rob Leurs
.
소스
International Journal of Molecular Sciences, Vol 25, Iss 9, p 5018 (2024)
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7 . Academic Journal
Synthesis and Pharmacological Characterization of New Photocaged Agonists for Histamine H3 and H4 Receptors
저자
by
Yang Zheng
;
Meichun Gao
;
Maikel Wijtmans
;
Henry F. Vischer
;
Rob Leurs
.
소스
Pharmaceuticals, Vol 17, Iss 4, p 536 (2024)
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7 . Academic Journal
Optical control of the β2-adrenergic receptor with opto-prop-2: A cis-active azobenzene analog of propranolol
저자
by
Reggie Bosma
;
Nicola C. Dijon
;
Yang Zheng
;
Hannes Schihada
;
Niels J. Hauwert
, et al.
소스
iScience, Vol 25, Iss 9, Pp 104882- (2022)
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7 . Academic Journal
Exploring the Effect of Cyclization of Histamine H1 Receptor Antagonists on Ligand Binding Kinetics
저자
by
Zhiyong Wang
;
Reggie Bosma
;
Sebastiaan Kuhne
;
Jelle van den Bor
;
Wrej Garabitian
, et al.
소스
ACS Omega, Vol 6, Iss 19, Pp 12755-12768 (2021)
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7 . Academic Journal
A toolbox of molecular photoswitches to modulate the CXCR3 chemokine receptor with light
저자
by
Xavier Gómez-Santacana
;
Sabrina M. de Munnik
;
Tamara A. M. Mocking
;
Niels J. Hauwert
;
Shanliang Sun
, et al.
소스
Beilstein Journal of Organic Chemistry, Vol 15, Iss 1, Pp 2509-2523 (2019)
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7 . Academic Journal
A NanoBRET-Based H3R Conformational Biosensor to Study Real-Time H3 Receptor Pharmacology in Cell Membranes and Living Cells
저자
by
Xiaoyuan Ma
;
Meichun Gao
;
Henry F. Vischer
;
Rob Leurs
.
소스
International Journal of Molecular Sciences, Vol 23, Iss 8211, p 8211 (2022)
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6 . Academic Journal
BRET-Based Biosensors to Measure Agonist Efficacies in Histamine H1 Receptor-Mediated G Protein Activation, Signaling and Interactions with GRKs and β-Arrestins
저자
by
Eléonore W. E. Verweij
;
Reggie Bosma
;
Meichun Gao
;
Jelle van den Bor
;
Betty Al Araaj
, et al.
소스
International Journal of Molecular Sciences, Vol 23, Iss 6, p 3184 (2022)
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7 . Academic Journal
Identification of TSPAN4 as Novel Histamine H4 Receptor Interactor
저자
by
Xiaoyuan Ma
;
Eléonore W. E. Verweij
;
Marco Siderius
;
Rob Leurs
;
Henry F. Vischer
.
소스
Biomolecules, Vol 11, Iss 8, p 1127 (2021)
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7 . Academic Journal
Analysis of Missense Variants in the Human Histamine Receptor Family Reveals Increased Constitutive Activity of E4106.30×30K Variant in the Histamine H1 Receptor
저자
by
Xiaoyuan Ma
;
Marta Arimont Segura
;
Barbara Zarzycka
;
Henry F. Vischer
;
Rob Leurs
.
소스
International Journal of Molecular Sciences, Vol 22, Iss 7, p 3702 (2021)
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