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1 . Academic Journal
Dependence on the Pyrimidine Biosynthetic Enzyme DHODH Is a Synthetic Lethal Vulnerability in Mutant KRAS-Driven Cancers
저자
by
Koundinya, Malvika
;
Sudhalter, Judith
;
Courjaud, Albane
;
Lionne, Bruno
;
Touyer, Gaetan
, et al.
소스
In
Cell Chemical Biology
21 June 2018 25(6):705-717
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7 . Academic Journal
A Robust Multiplex Mass Spectrometric Assay for Screening Small-Molecule Inhibitors of CD73 with Diverse Inhibition Modalities
저자
by
McManus, Jessica
;
He, Timothy
;
Gavigan, Julie-Ann
;
Marchand, Ghislaine
;
Vougier, Stephanie
, et al.
소스
In
SLAS Discovery
March 2018 23(3):264-273
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7 . Academic Journal
Small molecule activation of lecithin cholesterol acyltransferase modulates lipoprotein metabolism in mice and hamsters
저자
by
Chen, Zhu
;
Wang, Sheng-ping
;
Krsmanovic, Mihajlo L.
;
Castro-Perez, Jose
;
Gagen, Karen
, et al.
소스
In
Metabolism
April 2012 61(4):470-481
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7 . Academic Journal
Towards Prediction of In Vivo Intestinal Absorption Using a 96-Well Caco-2 Assay
저자
by
Skolnik, Suzanne
;
Lin, Xuena
;
Wang, Jianling
;
Chen, Xiao-Hui
;
He, Timothy
, et al.
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In
Journal of Pharmaceutical Sciences
July 2010 99(7):3246-3265
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7 . Academic Journal
Evaluation of Fluorescence- and Mass Spectrometry–Based CYP Inhibition Assays for Use in Drug Discovery
저자
by
Bell, Leslie
;
Bickford, Shari
;
Nguyen, Phong Hung
;
Wang, Jianling
;
He, Timothy
, et al.
소스
In
SLAS Discovery
June 2008 13(5):343-353
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7 . Academic Journal
A highly potent CD73 biparatopic antibody blocks organization of the enzyme active site through dual mechanisms.
저자
by
Stefano, James E.
;
Lord, Dana M.
;
Yanfeng Zhou
;
Jaworski, Julie
;
Hopke, Joern
, et al.
소스
Journal of Biological Chemistry
. 12/25/2020, Vol. 295 Issue 52, p18379-18389. 12p.
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7 . Academic Journal
Glutaminase is essential for the growth of triple-negative breast cancer cells with a deregulated glutamine metabolism pathway and its suppression synergizes with mTOR inhibition.
저자
by
Lampa, Michael
;
Arlt, Heike
;
He, Timothy
;
Ospina, Beatriz
;
Reeves, Jason
, et al.
소스
PLoS ONE
. 9/26/2017, Vol. 12 Issue 9, p1-24. 24p.
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7 . Academic Journal
Biomarkers profiling in patients with mucopolysaccharidosis and correlation with other primary biomarkers.
저자
by
An, Lin
;
Guo, Lilu
;
He, Timothy
;
Giugliani, Roberto
;
Zhao, Hongmei
, et al.
소스
Molecular Genetics & Metabolism
. Feb2023, Vol. 138 Issue 2, pN.PAG-N.PAG. 1p.
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7 . Academic Journal
Extreme Vulnerability of IDH1 Mutant Cancers to NAD+ Depletion.
저자
by
Tateishi, Kensuke
;
Wakimoto, Hiroaki
;
Iafrate, A. John
;
Tanaka, Shota
;
Loebel, Franziska
, et al.
소스
Cancer Cell
. Dec2015, Vol. 28 Issue 6, p773-784. 12p.
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7 . Academic Journal
Selective Inhibition of Mutant Isocitrate Dehydrogenase 1 (IDH1) via Disruption of a Metal Binding Network by an Allosteric Small Molecule.
저자
by
Gejing Deng
;
Junqing Shen
;
Ming Yin
;
McManus, Jessica
;
Mathie, Magali
, et al.
소스
Journal of Biological Chemistry
. 1/9/2015, Vol. 290 Issue 2, p762-774. 13p.
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