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1 . Academic Journal
TAK-861, a potent, orally available orexin receptor 2-selective agonist, produces wakefulness in monkeys and improves narcolepsy-like phenotypes in mouse models
저자
by
Kayo Mitsukawa
;
Michiko Terada
;
Ryuji Yamada
;
Taku Monjo
;
Tetsuaki Hiyoshi
, et al.
소스
Scientific Reports, Vol 14, Iss 1, Pp 1-15 (2024)
Open Access (DOAJ)
Scopus
Web of Science
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7 . Academic Journal
Effects of an OX2R agonist on migration and removal of tau from mouse brain
저자
by
Michiko Terada
;
Kayo Mitsukawa
;
Masanori Nakakariya
;
Tatsuki Koike
;
Haruhide Kimura
.
소스
Scientific Reports, Vol 14, Iss 1, Pp 1-12 (2024)
Open Access (DOAJ)
Scopus
Web of Science
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7 . Academic Journal
Orexin receptor 2 agonist activates diaphragm and genioglossus muscle through stimulating inspiratory neurons in the pre-Bötzinger complex, and phrenic and hypoglossal motoneurons in rodents.
저자
by
Ryuji Yamada
;
Tatsuki Koike
;
Masanori Nakakariya
;
Haruhide Kimura
.
소스
PLoS ONE, Vol 19, Iss 6, p e0306099 (2024)
Open Access (DOAJ)
Scopus
Web of Science
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6 . Academic Journal
Orexin 2 receptor (OX2R) protein distribution measured by autoradiography using radiolabeled OX2R-selective antagonist EMPA in rodent brain and peripheral tissues
저자
by
Kayo Mitsukawa
;
Haruhide Kimura
.
소스
Scientific Reports, Vol 12, Iss 1, Pp 1-13 (2022)
Open Access (DOAJ)
Scopus
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4 . Academic Journal
Strictly regulated agonist-dependent activation of AMPA-R is the key characteristic of TAK-653 for robust synaptic responses and cognitive improvement
저자
by
Atsushi Suzuki
;
Akiyoshi Kunugi
;
Yasukazu Tajima
;
Noriko Suzuki
;
Motohisa Suzuki
, et al.
소스
Scientific Reports, Vol 11, Iss 1, Pp 1-15 (2021)
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7 . Academic Journal
Inhibition of KDM1A activity restores adult neurogenesis and improves hippocampal memory in a mouse model of Kabuki syndrome
저자
by
Li Zhang
;
Genay Pilarowski
;
Emilio Merlo Pich
;
Atsushi Nakatani
;
John Dunlop
, et al.
소스
Molecular Therapy: Methods & Clinical Development, Vol 20, Iss , Pp 779-791 (2021)
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7 . Academic Journal
Author Correction: Strictly regulated agonist-dependent activation of AMPA-R is the key characteristic of TAK-653 for robust synaptic responses and cognitive improvement
저자
by
Atsushi Suzuki
;
Akiyoshi Kunugi
;
Yasukazu Tajima
;
Noriko Suzuki
;
Motohisa Suzuki
, et al.
소스
Scientific Reports, Vol 11, Iss 1, Pp 1-3 (2021)
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7 . Academic Journal
TAK-071, a novel M1 positive allosteric modulator with low cooperativity, improves cognitive function in rodents with few cholinergic side effects / 結合協調性の低いM1ポジティブアロステリックモジュレーターTAK-071は、げっ歯類でコリン作動性副作用を軽減しつつ優れた認知機能亢進作用を示す
저자
by
Haruhide Kimura
;
木村 温英
.
소스
Proceedings for Annual Meeting of The Japanese Pharmacological Society. 2020, :3-4
Open Access (JSTAGE)
Find it @ DONGA
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4 . Academic Journal
T‐495, a novel low cooperative M1 receptor positive allosteric modulator, improves memory deficits associated with cholinergic dysfunction and is characterized by low gastrointestinal side effect risk
저자
by
Takao Mandai
;
Yuu Sako
;
Emi Kurimoto
;
Yuji Shimizu
;
Minoru Nakamura
, et al.
소스
Pharmacology Research & Perspectives, Vol 8, Iss 1, Pp n/a-n/a (2020)
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7 . Academic Journal
TAK-071, a muscarinic M1 receptor positive allosteric modulator, attenuates scopolamine-induced quantitative electroencephalogram power spectral changes in cynomolgus monkeys.
저자
by
Emi Kurimoto
;
Masato Nakashima
;
Haruhide Kimura
;
Motohisa Suzuki
.
소스
PLoS ONE, Vol 14, Iss 3, p e0207969 (2019)
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