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1 . Academic Journal
Discovery and optimization of thiazole-based quorum sensing inhibitors as potent blockers of Pseudomonas aeruginosa pathogenicity
저자
by
Abdelsamie, Ahmed S.
;
Hamed, Mostafa M.
;
Schütz, Christian
;
Röhrig, Teresa
;
Kany, Andreas M.
, et al.
소스
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European Journal of Medicinal Chemistry
5 October 2024 276
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7 . Academic Journal
A hydrogel-based in vitro assay for the fast prediction of antibiotic accumulation in Gram-negative bacteria
저자
by
Richter, Robert
;
Kamal, Mohamed.A.M.
;
García-Rivera, Mariel A.
;
Kaspar, Jerome
;
Junk, Maximilian
, et al.
소스
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Materials Today Bio
September 2020 8
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7 . Academic Journal
Semisynthesis and biological evaluation of amidochelocardin derivatives as broad-spectrum antibiotics
저자
by
Grandclaudon, Charlotte
;
Birudukota, N.V. Suryanarayana
;
Elgaher, Walid A.M.
;
Jumde, Ravindra P.
;
Yahiaoui, Samir
, et al.
소스
In
European Journal of Medicinal Chemistry
15 February 2020 188
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7 . Academic Journal
Development of potential preclinical candidates with promising in vitro ADME profile for the inhibition of type 1 and type 2 17β-Hydroxysteroid dehydrogenases: Design, synthesis, and biological evaluation
저자
by
Abdelsamie, Ahmed S.
;
Salah, Mohamed
;
Siebenbürger, Lorenz
;
Hamed, Mostafa M.
;
Börger, Carsten
, et al.
소스
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European Journal of Medicinal Chemistry
15 September 2019 178:93-107
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7 . Academic Journal
Drifting of heme-coordinating group in imidazolylmethylxanthones leading to improved selective inhibition of CYP11B1
저자
by
Gobbi, Silvia
;
Hu, Qingzhong
;
Zimmer, Christina
;
Belluti, Federica
;
Rampa, Angela
, et al.
소스
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European Journal of Medicinal Chemistry
20 October 2017 139:60-67
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7 . Academic Journal
Pharmacological inhibition of protein kinase C (PKC)ζ downregulates the expression of cytokines involved in the pathogenesis of chronic obstructive pulmonary disease (COPD)
저자
by
Abdel-Halim, Mohammad
;
Darwish, Sarah S.
;
ElHady, Ahmed K.
;
Hoppstädter, Jessica
;
Abadi, Ashraf H.
, et al.
소스
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European Journal of Pharmaceutical Sciences
10 October 2016 93:405-409
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7 . Academic Journal
Systematic diversification of benzylidene heterocycles yields novel inhibitor scaffolds selective for Dyrk1A, Clk1 and CK2
저자
by
Mariano, Marica
;
Hartmann, Rolf W.
;
Engel, Matthias
.
소스
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European Journal of Medicinal Chemistry
13 April 2016 112:209-216
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5 . Academic Journal
Synthesis and biological evaluation of 3-tetrazolo steroidal analogs: Novel class of 5α-reductase inhibitors
저자
by
Aggarwal, Saurabh
;
Mahapatra, Manoj Kumar
;
Kumar, Rajnish
;
Bhardwaj, Tilak R.
;
Hartmann, Rolf W.
, et al.
소스
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Bioorganic & Medicinal Chemistry
15 February 2016 24(4):779-788
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7 . Academic Journal
Inhibition of aldosterone synthase (CYP11B2) by torasemide prevents atrial fibrosis and atrial fibrillation in mice
저자
by
Adam, Oliver
;
Zimmer, Christina
;
Hanke, Nina
;
Hartmann, Rolf W.
;
Klemmer, Birgit
, et al.
소스
In
Journal of Molecular and Cellular Cardiology
August 2015 85:140-150
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7 . Academic Journal
Identification of 4-(4-nitro-2-phenethoxyphenyl)pyridine as a promising new lead for discovering inhibitors of both human and rat 11β-Hydroxylase
저자
by
Hu, Qingzhong
;
Kunde, Jessica
;
Hanke, Nina
;
Hartmann, Rolf W.
.
소스
In
European Journal of Medicinal Chemistry
26 May 2015 96:139-150
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