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1 .
MK-8719, a Novel and Selective O-GlcNAcase Inhibitor That Reduces the Formation of Pathological Tau and Ameliorates Neurodegeneration in a Mouse Model of Tauopathy
저자
by
Giuseppe Terracina
;
Jerry P. Melchor
;
Cyrille Sur
;
David Kinsley
;
Lynn A. Hyde
, et al.
소스
Journal of Pharmacology and Experimental Therapeutics
. 374:252-263
Open Access (OpenAIRE)
Web of Science
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7 .
Discovery of MK-8719, a Potent O-GlcNAcase Inhibitor as a Potential Treatment for Tauopathies
저자
by
J. Fred Hess
;
Ramesh Kaul
;
Jacob Marcus
;
Jeanine E. Ballard
;
Joseph L. Duffy
, et al.
소스
Journal of medicinal chemistry
. 62(22)
Open Access (OpenAIRE)
Scopus
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7 . Academic Journal
Discovery and X-ray Crystallographic Analysis of a Spiropiperidine Iminohydantoin Inhibitor of β-Secretase.
저자
by
James C. Barrow
;
Shaun R. Stauffer
;
Kenneth E. Rittle
;
Phung L. Ngo
;
ZhiQiang Yang
, et al.
소스
Journal of Medicinal Chemistry
. Oct2008, Vol. 51 Issue 20, p6259-6262. 4p.
Full Text (ACS)
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7 .
Discovery of 6-(Fluoro-18F)-3-(1H-pyrrolo[2,3-c]pyridin-1-yl)isoquinolin-5-amine ([18F]-MK-6240): A Positron Emission Tomography (PET) Imaging Agent for Quantification of Neurofibrillary Tangles (NFTs)
저자
by
Patricia Miller
;
Yaode Wang
;
Joseph Della Rocca
;
Jeffrey L. Evelhoch
;
Paul J. Coleman
, et al.
소스
Journal of Medicinal Chemistry
. 59:4778-4789
Web of Science
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7 .
Inhibition of O-GlcNAcase leads to elevation of O-GlcNAc tau and reduction of tauopathy and cerebrospinal fluid tau in rTg4510 mice
저자
by
Julie Lee
;
Sherry X. Lu
;
Maureen Laverty
;
Brent D. Butts
;
Diane Grotz
, et al.
소스
Molecular Neurodegeneration
Molecular Neurodegeneration, Vol 12, Iss 1, Pp 1-16 (2017)
Open Access (BioMed Central)
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Scopus
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7 .
Insights into activity and inhibition from the crystal structure of human O-GlcNAcase
저자
by
Harold G. Selnick
;
Nathaniel L. Elsen
;
Sangita B. Patel
;
Dawn L. Hall
;
John C. Reid
, et al.
소스
Nature chemical biology
. 13(6)
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7 .
In Vivo Quantification of Calcitonin Gene-Related Peptide Receptor Occupancy by Telcagepant in Rhesus Monkey and Human Brain Using the Positron Emission Tomography Tracer [11C]MK-4232
저자
by
Harold G. Selnick
;
Mangay Williams
;
Patricia Miller
;
Guy Bormans
;
Hong Fan
, et al.
소스
Journal of Pharmacology and Experimental Therapeutics
. 347:478-486
Web of Science
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7 .
[11C]MK-4232: The First Positron Emission Tomography Tracer for the Calcitonin Gene-Related Peptide Receptor
저자
by
Samuel L. Graham
;
Joseph G. Bruno
;
Scott D. Mosser
;
Harold G. Selnick
;
Sandra M. Sanabria-Bohórquez
, et al.
소스
ACS Medicinal Chemistry Letters
. 4:863-868
Open Access (OpenAIRE)
Web of Science
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7 .
O2‐13‐04: Early Clinical Results and Preclinical Validation of the O‐Glcnacase (OGA) Inhibitor Mk‐8719 as a Novel Therapeutic for the Treatment of Tauopathies
저자
by
Jacob Marcus
;
Ruben Declercq
;
Mali Cosden
;
Cristian Salinas
;
John J. Renger
, et al.
소스
Alzheimer's & Dementia
. 12
Scopus
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7 .
MK-8825: A potent and selective CGRP receptor antagonist with good oral activity in rats
저자
by
Samuel L. Graham
;
Christine Fandozzi
;
Eric L. Moore
;
Donnette D. Staas
;
Ian M. Bell
, et al.
소스
Bioorganic & Medicinal Chemistry Letters
. 22:3941-3945
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