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1 . Academic Journal
Identification and evaluation of small-molecule inhibitors against the dNTPase SAMHD1 via a comprehensive screening funnel
저자
by
Si Min Zhang
;
Cynthia B.J. Paulin
;
Huazhang Shu
;
Miriam Yagüe-Capilla
;
Maurice Michel
, et al.
소스
iScience, Vol 27, Iss 2, Pp 108907- (2024)
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7 . Academic Journal
Ribonucleotide reductase inhibitors suppress SAMHD1 ara‐CTPase activity enhancing cytarabine efficacy
저자
by
Sean G Rudd
;
Nikolaos Tsesmetzis
;
Kumar Sanjiv
;
Cynthia BJ Paulin
;
Lakshmi Sandhow
, et al.
소스
EMBO Molecular Medicine, Vol 12, Iss 3, Pp n/a-n/a (2020)
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7 . Academic Journal
Targeted NUDT5 inhibitors block hormone signaling in breast cancer cells
저자
by
Brent D. G. Page
;
Nicholas C. K. Valerie
;
Roni H. G. Wright
;
Olov Wallner
;
Rebecka Isaksson
, et al.
소스
Nature Communications, Vol 9, Iss 1, Pp 1-14 (2018)
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7 . Academic Journal
CETSA screening identifies known and novel thymidylate synthase inhibitors and slow intracellular activation of 5-fluorouracil
저자
by
Helena Almqvist
;
Hanna Axelsson
;
Rozbeh Jafari
;
Chen Dan
;
André Mateus
, et al.
소스
Nature Communications, Vol 7, Iss 1, Pp 1-11 (2016)
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7 . Academic Journal
Author Correction: Targeted NUDT5 inhibitors block hormone signaling in breast cancer cells
저자
by
Brent D. G. Page
;
Nicholas C. K. Valerie
;
Roni H. G. Wright
;
Olov Wallner
;
Rebecka Isaksson
, et al.
소스
Nature Communications, Vol 10, Iss 1, Pp 1-1 (2019)
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7 . Academic Journal
Crystal structures of the kinase domain of the sulfate-activating complex in Mycobacterium tuberculosis.
저자
by
Ömer Poyraz
;
Katharina Brunner
;
Bernhard Lohkamp
;
Hanna Axelsson
;
Lars G J Hammarström
, et al.
소스
PLoS ONE, Vol 10, Iss 3, p e0121494 (2015)
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7 . Academic Journal
Using High Content Imaging to Quantify Target Engagement in Adherent Cells
저자
by
Hanna Axelsson, author
;
Helena Almqvist, author
;
Brinton Seashore-Ludlow, author
.
소스
Journal of Visualized Experiments
. (141)
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5 .
Subcellular mapping of the protein landscape of SARS-CoV-2 infected cells for target-centric drug repurposing
저자
by
Jayasankar Mohanakrishnan Kaimal
;
Marianna Tampere
;
Trang H. Le
;
Ulrika Axelsson
;
Hao Xu
, et al.
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7 .
Development of a chemical probe against NUDT15
저자
by
Saeed Eshtad
;
Ingrid Almlöf
;
Pål Stenmark
;
Matthieu Desroses
;
Armando Cázares-Körner
, et al.
소스
Nature chemical biology
Nature Chemical Biology
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7 .
Quantitative Interpretation of Intracellular Drug Binding and Kinetics Using the Cellular Thermal Shift Assay
저자
by
Brinton Seashore-Ludlow
;
Helena Almqvist
;
Mats Jonsson
;
Thomas Lundbäck
;
Björn Dahlgren
, et al.
소스
Biochemistry
. 57:6715-6725
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