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1 . Academic Journal
Design and synthesis of fused azacyclic and azaspirocyclic γ-lactams targeting dopaminergic D2/D4 receptors
저자
by
Lalut, Julien
;
Hocine, Sofiane
;
Maertens, Gaëtan
;
Vilchis-Reyes, Miguel
;
Hanessian, Stephen
.
소스
In
Journal of Molecular Structure
5 March 2024 1299
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7 . Academic Journal
Revisiting the dipeptidyl carboxypeptidase inhibitor captopril as a source of pan anti-trypanosomatid agents
저자
by
Garsi, Jean-Baptiste
;
Hocine, Sofiane
;
Hensienne, Raphaël
;
Moitessier, Matthieu
;
Denton, Helen
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 September 2024 110
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7 . Academic Journal
1,2- trans -Diaminocyclohexane (DACH) in Asymmetric Catalysis: Nearing Fifty Years of Faithful Service and Counting.
저자
by
Mishra, Akash
;
Hanessian, Stephen
.
소스
Synthesis
. Sep2024, Vol. 56 Issue 18, p2747-2885. 139p.
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4 . Academic Journal
My 50-Plus Years of Academic Research Collaborations with Industry. A Retrospective.
저자
by
Hanessian, Stephen
.
소스
Journal of Organic Chemistry; 7/5/2024, Vol. 89 Issue 13, p9147-9186, 40p
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3 . Academic Journal
In search of constrained FTY720 and phytosphingosine analogs as dual acting anticancer agents targeting metabolic and epigenetic pathways
저자
by
Garsi, Jean-Baptiste
;
Sernissi, Lorenzo
;
Vece, Vito
;
Hanessian, Stephen
;
McCracken, Alison N.
, et al.
소스
In
European Journal of Medicinal Chemistry
5 November 2018 159:217-242
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7 . Academic Journal
Design and synthesis of novel N-sulfonyl-2-indoles that behave as 5-HT6 receptor ligands with significant selectivity for D3 over D2 receptors
저자
by
Saavedra, Oscar M.
;
Karila, Delphine
;
Brossard, Dominique
;
Rojas, Anne
;
Dupuis, Delphine
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 January 2017 25(1):38-52
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7 . Academic Journal
Towards combining backbone and sugar constraint in 3′-3′ bis-phosphonate tethered 2′-4′ bridged LNA oligonucleotide trimers.
저자
by
Duchamp, Edouard
;
Vasquez, Guillermo
;
Firoozi, Neda
;
Freestone, Graeme C.
;
Oestergaard, Michael
, et al.
소스
RSC Advances; 2024, Vol. 14 Issue 33, p23583-23591, 9p
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7 . Academic Journal
Pseudodiproline (Pro–Cyp) Oligomers Fold into Helical Polyproline Type secondary structures.
저자
by
Garsi, Jean-Baptiste
;
Aguiar, Pedro M.
;
Berger, Gilles
;
Maris, Thierry
;
Hanessian, Stephen
.
소스
Journal of Organic Chemistry; 4/5/2024, Vol. 89 Issue 7, p4283-4293, 11p
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7 . Academic Journal
Effects of stereochemistry, saturation, and hydrocarbon chain length on the ability of synthetic constrained azacyclic sphingolipids to trigger nutrient transporter down-regulation, vacuolation, and cell death
저자
by
Perryman, Michael S.
;
Tessier, Jérémie
;
Wiher, Timothy
;
O’Donoghue, Heather
;
McCracken, Alison N.
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 September 2016 24(18):4390-4397
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7 . Academic Journal
Synthesis and biological evaluation of sialyl-oligonucleotide conjugates targeting leukocyte B trans-membranal receptor CD22 as delivery agents for nucleic acid drugs
저자
by
St-Pierre, Gabrielle
;
Pal, Sudip
;
Østergaard, Michael E.
;
Zhou, Tianyuan
;
Yu, Jinghua
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 June 2016 24(11):2397-2409
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