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1 . Academic Journal
Machine Learning ADME Models in Practice: Four Guidelines from a Successful Lead Optimization Case Study.
저자
by
Rich, Alexander S.
;
Chan, Yvonne H.
;
Birnbaum, Benjamin
;
Haider, Kamran
;
Haimson, Joshua
, et al.
소스
ACS Medicinal Chemistry Letters; 8/8/2024, Vol. 15 Issue 8, p1169-1173, 5p
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7 . Academic Journal
Repurposing a Histamine Detection Platform for High-Throughput Screening of Histidine Decarboxylase
저자
by
Juang, Yu-Chi
;
Fradera, Xavier
;
Han, Yongxin
;
Partridge, Anthony William
.
소스
In
SLAS Discovery
October 2018 23(9):974-981
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6 . Academic Journal
Discovery of IDO1 inhibitors containing a decahydroquinoline, decahydro-1,6-naphthyridine, or octahydro-1H-pyrrolo[3,2-c]pyridine scaffold
저자
by
Yu, Wensheng
;
Deng, Yongqi
;
Sloman, David
;
Li, Derun
;
Liu, Kun
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 October 2021 49
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7 . Academic Journal
SAR towards indoline and 3-azaindoline classes of IDO1 inhibitors
저자
by
Yu, Wensheng
;
Deng, Yongqi
;
Hopkins, Brett
;
Huang, Xianhai
;
Sloman, David
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 September 2021 47
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7 . Academic Journal
Discovery of MK-8768, a Potent and Selective mGluR2 Negative Allosteric Modulator.
저자
by
Rudd, Michael T.
;
Manley, Peter J.
;
Hanney, Barbara
;
Meng, Zhaoyang
;
Shu, Youheng
, et al.
소스
ACS Medicinal Chemistry Letters; 8/10/2023, Vol. 14 Issue 8, p1088-1094, 7p
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7 . Academic Journal
Correlating the fractional inhibition of caspase-3 in NT2 cells with apoptotic markers using an active-caspase-3 enzyme-linked immunosorbent assay
저자
by
Tawa, Paul
;
Giroux, Andre
;
Grimm, Erich
;
Han, Yongxin
;
Nicholson, Donald W.
, et al.
소스
In
Analytical Biochemistry
2006 350(1):32-40
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7 . Academic Journal
WNT5B promotes vascular smooth muscle cell dedifferentiation via mitochondrial dynamics regulation in chronic thromboembolic pulmonary hypertension.
저자
by
Wang, Feng
;
Zhen, Yanan
;
Si, Chaozeng
;
Wang, Cheng
;
Pan, Lin
, et al.
소스
Journal of Cellular Physiology
. Jan2022, Vol. 237 Issue 1, p789-803. 15p.
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7 . Academic Journal
Solid phase parallel synthesis of highly substituted thiophene derivatives and identification of novel phosphodiesterase-4 (PDE-4) inhibitors
저자
by
Han, Yongxin
;
Giroux, André
;
Lépine, Carole
;
Laliberté, France
;
Huang, Zheng
, et al.
소스
In
Tetrahedron
1999 55(39):11669-11685
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7 . Academic Journal
Role of pyroptosis in atherosclerosis and its therapeutic implications.
저자
by
He, Bin
;
Nie, Qiangqiang
;
Wang, Feng
;
Han, Yongxin
;
Yang, Bo
, et al.
소스
Journal of Cellular Physiology
. Oct2021, Vol. 236 Issue 10, p7159-7175. 17p.
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7 . Periodical
Oxetane Promise Delivered: Discovery of Long-Acting IDO1 Inhibitors Suitable for Q3W Oral or Parenteral Dosing
저자
by
Li, Derun
;
Sloman, David L.
;
Achab, Abdelghani
;
Zhou, Hua
;
McGowan, Meredeth A.
, et al.
소스
Journal of Medicinal Chemistry; April 2022, Vol. 65 Issue: 8 p6001-6016, 16p
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