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1 . Academic Journal
Safety, tolerability, pharmacokinetics, and antimalarial efficacy of a novel Plasmodium falciparum ATP4 inhibitor SJ733: a first-in-human and induced blood-stage malaria phase 1a/b trial
저자
by
Gaur, Aditya H
;
McCarthy, James S
;
Panetta, John C
;
Dallas, Ronald H
;
Woodford, John
, et al.
소스
In
The Lancet Infectious Diseases
August 2020 20(8):964-975
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7 . Academic Journal
A Phase 1, Randomized, Double‐Blind, Placebo‐Controlled, Single Ascending Dose Trial of AWZ1066S, an Anti‐Wolbachia Candidate Macrofilaricide.
저자
by
Devereux, Graham
;
Bula, Marcin
;
Tripp, Karen
;
Fitzgerald, Richard
;
Eraut, Nicola
, et al.
소스
Clinical Pharmacology in Drug Development
. Sep2024, Vol. 13 Issue 9, p1071-1081. 11p.
Scopus
Find it @ DONGA
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7 . Periodical
A Phase 1, Randomized, Double‐Blind, Placebo‐Controlled, Single Ascending Dose Trial of AWZ1066S, an Anti‐WolbachiaCandidate Macrofilaricide
저자
by
Devereux, Graham
;
Bula, Marcin
;
Tripp, Karen
;
Fitzgerald, Richard
;
Eraut, Nicola
, et al.
소스
Clinical Pharmacology in Drug Development; September 2024, Vol. 13 Issue: 9 p1071-1081, 11p
Web of Science
Scopus
JCR 저널정보
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7 . Academic Journal
A simple fluorescence-based assay for quantification of the Toll-Like Receptor agonist E6020 in vaccine formulations
저자
by
Pollet, Jeroen
;
Versteeg, Leroy
;
Rezende, Wanderson
;
Strych, Ulrich
;
Gusovsky, Fabian
, et al.
소스
In
Vaccine
7 March 2017 35(10):1410-1416
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7 . Academic Journal
Combinations of the azaquinazoline anti-Wolbachia agent, AWZ1066S, with benzimidazole anthelmintics synergise to mediate sub-seven-day sterilising and curative efficacies in experimental models of filariasis.
저자
by
Hegde, Shrilakshmi
;
Marriott, Amy E.
;
Pionnier, Nicolas
;
Steven, Andrew
;
Bulman, Christina
, et al.
소스
Frontiers in Microbiology; 2024, p1-17, 17p
Web of Science
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7 . Academic Journal
The impact of vaccine-linked chemotherapy on liver health in a mouse model of chronic Trypanosoma cruzi infection.
저자
by
Nguyen, Duc Minh
;
Poveda, Cristina
;
Pollet, Jeroen
;
Gusovsky, Fabian
;
Bottazzi, Maria Elena
, et al.
소스
PLoS Neglected Tropical Diseases
. 11/21/2023, Vol. 17 Issue 11, p1-18. 18p.
Scopus
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7 . Academic Journal
Vaccine-linked chemotherapy improves cardiac structure and function in a mouse model of chronic Chagas disease.
저자
by
Jones, Kathryn M.
;
Mangin, Elise N.
;
Reynolds, Corey L.
;
Villanueva, Liliana E.
;
Vladimir Cruz, Julio
, et al.
소스
Frontiers in Cellular & Infection Microbiology; 2/9/2023, Vol. 13, p1-18, 18p
Web of Science
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7 . Academic Journal
Transformation of the Manufacturing Process from Discovery to Kilogram Scale for AWZ1066S: A Highly Specific Anti-Wolbachia Drug Candidate for a Short-Course Treatment of Filariasis.
저자
by
Hong, W. David
;
O'Neill, Paul M.
;
Taylor, Mark J.
;
Turner, Joseph D.
;
Ward, Stephen A.
, et al.
소스
Organic Process Research & Development; 1/20/2023, Vol. 27 Issue 1, p42-53, 12p
Full Text (ACS)
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7 . Academic Journal
Vaccine-linked chemotherapy with a low dose of benznidazole plus a bivalent recombinant protein vaccine prevents the development of cardiac fibrosis caused by Trypanosoma cruzi in chronically-infected BALB/c mice.
저자
by
Dzul-Huchim, Victor Manuel
;
Ramirez-Sierra, Maria Jesus
;
Martinez-Vega, Pedro Pablo
;
Rosado-Vallado, Miguel Enrique
;
Arana-Argaez, Victor Ermilo
, et al.
소스
PLoS Neglected Tropical Diseases
. 9/12/2022, Vol. 16 Issue 9, p1-20. 20p.
Scopus
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7 . Academic Journal
Crystallization-Based Synthetic Route to Antimalarial Agent BRD5018: Diazocene Ring Formation via a Staudinger-aza-Wittig Reaction on an Azetidine-Ribose Template.
저자
by
Mitasev, Branko
;
Jiong Yang
;
Gusovsky, Fabian
;
Girish, Dixit
;
Khile, Anil Shahaji
, et al.
소스
Organic Process Research & Development; 3/18/2022, Vol. 26 Issue 3, p817-831, 15p
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