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1 .
TRPV4 Specific Inhibition Ameliorates Fluid-Induced Lung Injury
저자
by
Shailesh Bihari
;
Melissa H. Costell
;
Tara Bouchier
;
David J. Behm
;
Mark Burgert
, et al.
소스
SSRN Electronic Journal
.
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7 .
Discovery of GSK2798745: A Clinical Candidate for Inhibition of Transient Receptor Potential Vanilloid 4 (TRPV4)
저자
by
Eidam Hilary Schenck
;
Theresa J. Roethke
;
Linda S. Barton
;
Fox Ryan Michael
;
Steve Zhao
, et al.
소스
ACS Med Chem Lett
Open Access (OpenAIRE)
Web of Science
Scopus
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7 .
Design and Optimization of an Acyclic Amine Series of TRPV4 Antagonists by Electronic Modulation of Hydrogen Bond Interactions
저자
by
Guosen Ye
;
Arthur Shu
;
Dennis A. Holt
;
Patrick Stoy
;
Carla A. Donatelli
, et al.
소스
Journal of medicinal chemistry
. 63(23)
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7 . Academic Journal
TRPV4 inhibition counteracts edema and inflammation and improves pulmonary function and oxygen saturation in chemically induced acute lung injury.
저자
by
Balakrishna, Shrilatha
;
Weifeng Song
;
Achanta, Satyanarayana
;
Doran, Stephen F.
;
Liu, Boyi
, et al.
소스
American Journal of Physiology: Lung Cellular & Molecular Physiology
. 2014, Vol. 307 Issue 2, pL158-L172. 15p.
Web of Science
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7 .
Reverse Hydroxamate Inhibitors of Bone Morphogenetic Protein 1
저자
by
Theresa J. Roethke
;
Guosen Ye
;
Hong Zhang
;
Robert T. Gampe
;
Robert A. Reid
, et al.
소스
ACS Medicinal Chemistry Letters
. 9:736-740
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7 . Academic Journal
Discovery of Aminofurazan-azabenzimidazoles as Inhibitors of Rho-Kinase with High Kinase Selectivity and Antihypertensive Activity.
저자
by
Robert A. Stavenger
;
Haifeng Cui
;
Sarah E. Dowdell
;
Robert G. Franz
;
Dimitri E. Gaitanopoulos
, et al.
소스
Journal of Medicinal Chemistry
. Jan2007, Vol. 50 Issue 1, p2-5. 4p.
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7 . Academic Journal
Development of Dihydropyridone Indazole Amides as Selective Rho-Kinase Inhibitors.
저자
by
Krista B. Goodman
;
Haifeng Cui
;
Sarah E. Dowdell
;
Dimitri E. Gaitanopoulos
;
Robert L. Ivy
, et al.
소스
Journal of Medicinal Chemistry
. Jan2007, Vol. 50 Issue 1, p6-9. 4p.
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7 .
Discovery of GSK2193874: An Orally Active, Potent, and Selective Blocker of Transient Receptor Potential Vanilloid 4
저자
by
Theresa J. Roethke
;
Weike Bao
;
Dennis A. Holt
;
David J. Behm
;
Eidam Hilary Schenck
, et al.
소스
ACS Medicinal Chemistry Letters
. 8:549-554
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7 .
Discovery of Pyrrolidine Sulfonamides as Selective and Orally Bioavailable Antagonists of Transient Receptor Potential Vanilloid-4 (TRPV4)
저자
by
Arthur Shu
;
Carla A. Donatelli
;
Sanchez Robert
;
Melissa H. Costell
;
Carl Brooks
, et al.
소스
Journal of medicinal chemistry
. 61(21)
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7 .
Design of amidobenzimidazole STING receptor agonists with systemic activity
저자
by
Joshi M. Ramanjulu
;
G. Scott Pesiridis
;
Jingsong Yang
;
Nestor Concha
;
Robert Singhaus
, et al.
소스
Nature
. 564(7736)
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