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1 . Academic Journal
Sulfonylpiperidines as novel, antibacterial inhibitors of Gram-positive thymidylate kinase (TMK)
저자
by
Martínez-Botella, Gabriel
;
Loch, James T.
;
Green, Oluyinka M.
;
Kawatkar, Sameer P.
;
Olivier, Nelson B.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 January 2013 23(1):169-173
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7 . Academic Journal
Inhibitors of the acetyltransferase domain of N-acetylglucosamine-1-phosphate-uridylyltransferase/glucosamine-1-phosphate-acetyltransferase (GlmU). Part 2: Optimization of physical properties leading to antibacterial aryl sulfonamides
저자
by
Stokes, Suzanne S.
;
Albert, Robert
;
Buurman, Ed T.
;
Andrews, Beth
;
Shapiro, Adam B.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 December 2012 22(23):7019-7023
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7 . Academic Journal
Inhibitors of acetyltransferase domain of N-acetylglucosamine-1-phosphate-uridyltransferase/glucosamine-1-phosphate-acetyltransferase (GlmU). Part 1: Hit to lead evaluation of a novel arylsulfonamide series
저자
by
Green, Oluyinka M.
;
McKenzie, Andrew R.
;
Shapiro, Adam B.
;
Otterbein, Ludovic
;
Ni, Haihong
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 February 2012 22(4):1510-1519
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7 . Academic Journal
Antibacterial Inhibitors ofGram-Positive ThymidylateKinase: Structure–Activity Relationships and Chiral Preferenceof a New Hydrophobic Binding Region.
저자
by
Kawatkar, Sameer P.
;
Keating, Thomas A.
;
Olivier, Nelson B.
;
Breen, John N.
;
Green, Oluyinka M.
, et al.
소스
Journal of Medicinal Chemistry
. Jun2014, Vol. 57 Issue 11, p4584-4597. 14p.
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7 . Periodical
In VivoValidation of Thymidylate Kinase (TMK) with a Rationally Designed, Selective Antibacterial Compound
저자
by
Keating, Thomas A.
;
Newman, Joseph V.
;
Olivier, Nelson B.
;
Otterson, Linda G.
;
Andrews, Beth
, et al.
소스
ACS Chemical Biology; November 2012, Vol. 7 Issue: 11 p1866-1872, 7p
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7 . Academic Journal
Discovery of Selective and Potent Inhibitors of Gram-Positive Bacterial Thymidylate Kinase (TMK)
저자
by
Martinez-Botella, Gabriel
;
Breen, John N.
;
Duffy, James E. S.
;
Dumas, Jacques
;
Geng, Bolin
, et al.
소스
JOURNAL OF MEDICINAL CHEMISTRY
; NOV 22 2012, 55 22, p10010-p10021, 12p.
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7 . Academic Journal
In Vivo Validation of Thymidylate Kinase (TMK) with a Rationally Designed, Selective Antibacterial Compound
저자
by
Keating, Thomas A.
;
Newman, Joseph V.
;
Olivier, Nelson B.
;
Otterson, Linda G.
;
Andrews, Beth
, et al.
소스
ACS CHEMICAL BIOLOGY
; NOV 2012, 7 11, p1866-p1872, 7p.
Full Text (ACS)
Scopus
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