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1 . Academic Journal
From virtual screening hits targeting a cryptic pocket in BACE-1 to a nontoxic brain permeable multitarget anti-Alzheimer lead with disease-modifying and cognition-enhancing effects
저자
by
Pont, Caterina
;
Ginex, Tiziana
;
Griñán-Ferré, Christian
;
Scheiner, Matthias
;
Mattellone, Alexia
, et al.
소스
In
European Journal of Medicinal Chemistry
5 December 2021 225
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7 . Academic Journal
Potential pharmacological strategies targeting the Niemann-Pick C1 receptor and Ebola virus glycoprotein interaction
저자
by
Morales-Tenorio, Marcos
;
Ginex, Tiziana
;
Cuesta-Geijo, Miguel Ángel
;
Campillo, Nuria E.
;
Muñoz-Fontela, César
, et al.
소스
In
European Journal of Medicinal Chemistry
5 November 2021 223
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7 . Academic Journal
N-benzyl 4,4-disubstituted piperidines as a potent class of influenza H1N1 virus inhibitors showing a novel mechanism of hemagglutinin fusion peptide interaction
저자
by
de Castro, Sonia
;
Ginex, Tiziana
;
Vanderlinden, Evelien
;
Laporte, Manon
;
Stevaert, Annelies
, et al.
소스
In
European Journal of Medicinal Chemistry
15 May 2020 194
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7 . Academic Journal
Pharmacology and preclinical validation of a novel anticancer compound targeting PEPCK-M
저자
by
Aragó, Marc
;
Moreno-Felici, Juan
;
Abás, Sonia
;
Rodríguez-Arévalo, Sergio
;
Hyroššová, Petra
, et al.
소스
In
Biomedicine & Pharmacotherapy
January 2020 121
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7 . Academic Journal
Potential of aryl–urea–benzofuranylthiazoles hybrids as multitasking agents in Alzheimer's disease
저자
by
Kurt, Belma Zengin
;
Gazioglu, Isil
;
Basile, Livia
;
Sonmez, Fatih
;
Ginex, Tiziana
, et al.
소스
In
European Journal of Medicinal Chemistry
18 September 2015 102:80-92
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7 . Academic Journal
MBC and ECBL libraries: outstanding tools for drug discovery.
저자
by
Ginex, Tiziana
;
Madruga, Enrique
;
Martinez, Ana
;
Gil, Carmen
.
소스
Frontiers in Pharmacology; 2023, p1-12, 12p
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6 . Academic Journal
Screening and Biological Evaluation of Soluble Epoxide Hydrolase Inhibitors: Assessing the Role of Hydrophobicity in the Pharmacophore-Guided Search of Novel Hits.
저자
by
Vázquez, Javier
;
Ginex, Tiziana
;
Herrero, Albert
;
Morisseau, Christophe
;
Hammock, Bruce D.
, et al.
소스
Journal of Chemical Information & Modeling; 5/22/2023, Vol. 63 Issue 10, p3209-3225, 17p
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7 . Academic Journal
N′‑Phenylacetohydrazide Derivatives as Potent Ebola Virus Entry Inhibitors with an Improved Pharmacokinetic Profile.
저자
by
Garcia-Rubia, Alfonso
;
Lasala, Fátima
;
Ginex, Tiziana
;
Morales-Tenorio, Marcos
;
Olal, Catherine
, et al.
소스
Journal of Medicinal Chemistry; 4/27/2023, Vol. 66 Issue 8, p5465-5483, 19p
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7 . Academic Journal
Inhibition of β‑Amyloid Aggregation in Alzheimer's Disease: The Key Role of (Pro)electrophilic Warheads.
저자
by
Basagni, Filippo
;
Naldi, Marina
;
Ginex, Tiziana
;
Luque, F. Javier
;
Fagiani, Francesca
, et al.
소스
ACS Medicinal Chemistry Letters; 11/10/2022, Vol. 13 Issue 11, p1812-1818, 7p
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7 . Academic Journal
The structural role of SARS-CoV-2 genetic background in the emergence and success of spike mutations: The case of the spike A222V mutation.
저자
by
Ginex, Tiziana
;
Marco-Marín, Clara
;
Wieczór, Miłosz
;
Mata, Carlos P.
;
Krieger, James
, et al.
소스
PLoS Pathogens
. 7/11/2022, Vol. 18 Issue 7, p1-28. 28p.
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