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1 . Academic Journal
Fragment-based and structure-guided discovery of perforin inhibitors
저자
by
Jose, Jiney
;
Law, Ruby H.P.
;
Leung, Eleanor W.W.
;
Wai, Dorothy C.C.
;
Akhlaghi, Hedieh
, et al.
소스
In
European Journal of Medicinal Chemistry
5 December 2023 261
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7 . Academic Journal
Synthesis and biological evaluation of sulfonamide analogues of the phosphatidylinositol 3-kinase inhibitor ZSTK474
저자
by
Gamage, Swarna A.
;
Giddens, Anna C.
;
Tsang, Kit Y.
;
Flanagan, Jack U.
;
Kendall, Jackie D.
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 October 2017 25(20):5859-5874
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7 . Academic Journal
Analogues of DNA minor groove cross-linking agents incorporating aminoCBI, an amino derivative of the duocarmycins: Synthesis, cytotoxicity, and potential as payloads for antibody–drug conjugates
저자
by
Giddens, Anna C.
;
Lee, Ho H.
;
Lu, Guo-Liang
;
Miller, Christian K.
;
Guo, Jun
, et al.
소스
In
Bioorganic & Medicinal Chemistry
15 November 2016 24(22):6075-6081
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7 . Academic Journal
Synthetic studies towards isomeric pyrazolopyrimidines as potential ATP synthesis inhibitors of Mycobacterium tuberculosis. Structural correction of reported N-(6-(2-(dimethylamino)ethoxy)-5-fluoropyridin-3-yl)-2-(4-fluorophenyl)-5-(trifluoromethyl)pyrazolo[1,5-α]pyrimidin-7-amine
저자
by
Choi, Peter J.
;
Lu, Guo-Liang
;
Sutherland, Hamish S.
;
Giddens, Anna C.
;
Franzblau, Scott G.
, et al.
소스
In
Tetrahedron Letters
2 February 2022 90
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7 . Academic Journal
Semi-synthesis of bioactive fluorescent analogues of the cytotoxic marine alkaloid discorhabdin C
저자
by
Lam, Cary F.C.
;
Giddens, Anna C.
;
Chand, Natasha
;
Webb, Victoria L.
;
Copp, Brent R.
.
소스
In
Tetrahedron
15 April 2012 68(15):3187-3194
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7 . Academic Journal
Novel pyrazolo[1,5-a]pyridines as p110α-selective PI3 kinase inhibitors: Exploring the benzenesulfonohydrazide SAR
저자
by
Kendall, Jackie D.
;
Giddens, Anna C.
;
Tsang, Kit Yee
;
Frédérick, Raphaël
;
Marshall, Elaine S.
, et al.
소스
In
Bioorganic & Medicinal Chemistry
1 January 2012 20(1):58-68
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7 . Academic Journal
Natural product inhibitors of fatty acid biosynthesis: synthesis of the marine microbial metabolites pseudopyronines A and B and evaluation of their anti-infective activities
저자
by
Giddens, Anna C.
;
Nielsen, Lone
;
Boshoff, Helena I.
;
Tasdemir, Deniz
;
Perozzo, Remo
, et al.
소스
In
Tetrahedron
2008 64(7):1242-1249
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7 . Academic Journal
Synthesis and Structure–Activity Relationships for the Anti-Mycobacterial Activity of 3-Phenyl- N -(Pyridin-2-ylmethyl)Pyrazolo[1,5- a ]Pyrimidin-7-Amines.
저자
by
Sutherland, Hamish S.
;
Choi, Peter J.
;
Lu, Guo-Liang
;
Giddens, Anna C.
;
Tong, Amy S. T.
, et al.
소스
Pharmaceuticals (14248247)
. Sep2022, Vol. 15 Issue 9, pN.PAG-N.PAG. 31p.
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7 . Academic Journal
Novel pyrazolo[1,5-a]pyridines with improved aqueous solubility as p110α-selective PI3 kinase inhibitors
저자
by
Kendall, Jackie D.
;
Giddens, Anna C.
;
Tsang, Kit Yee
;
Marshall, Elaine S.
;
Lill, Claire L.
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 January 2017 27(2):187-190
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7 . Periodical
Inhibition of the Cytolytic Protein Perforin Prevents Rejection of Transplanted Bone Marrow Stem Cells in Vivo
저자
by
Spicer, Julie A.
;
Miller, Christian K.
;
O’Connor, Patrick D.
;
Jose, Jiney
;
Giddens, Anna C.
, et al.
소스
Journal of Medicinal Chemistry; March 2020, Vol. 63 Issue: 5 p2229-2239, 11p
Full Text (ACS)
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