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1 . Academic Journal
Robust Prediction of Relative Binding Energies for Protein–Protein Complex Mutations Using Free Energy Perturbation Calculations
저자
by
Sampson, Jared M.
;
Cannon, Daniel A.
;
Duan, Jianxin
;
Epstein, Jordan C.K.
;
Sergeeva, Alina P.
, et al.
소스
In
Journal of Molecular Biology
15 August 2024 436(16)
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7 . Academic Journal
Regenerable Biosensors for Small-Molecule Kinetic Characterization Using SPR
저자
by
Gunnarsson, Anders
;
Stubbs, Christopher J.
;
Rawlins, Philip B.
;
Taylor-Newman, Eleanor
;
Lee, Wei-chao
, et al.
소스
In
SLAS Discovery
June 2021 26(5):730-739
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7 . Academic Journal
Agonists and Antagonists of Protease-Activated Receptor 2 Discovered within a DNA-Encoded Chemical Library Using Mutational Stabilization of the Target
저자
by
Brown, Dean G.
;
Brown, Giles A.
;
Centrella, Paolo
;
Certel, Kaan
;
Cooke, Robert M.
, et al.
소스
In
SLAS Discovery
June 2018 23(5):429-436
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7 . Academic Journal
Direct cell extraction of membrane proteins for structure–function analysis.
저자
by
Drulyte, Ieva
;
Gutgsell, Aspen Rene
;
Lloris-Garcerá, Pilar
;
Liss, Michael
;
Geschwindner, Stefan
, et al.
소스
Scientific Reports
. 1/25/2023, Vol. 13 Issue 1, p1-8. 8p.
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7 . Academic Journal
Fragment-assisted hit investigation involving integrated HTS and fragment screening: Application to the identification of phosphodiesterase 10A (PDE10A) inhibitors
저자
by
Varnes, Jeffrey G.
;
Geschwindner, Stefan
;
Holmquist, Christopher R.
;
Forst, Janet
;
Wang, Xia
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
1 January 2016 26(1):197-202
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7 . Academic Journal
Importance of Binding Site Hydration and Flexibility Revealed When Optimizing a Macrocyclic Inhibitor of the Keap1-Nrf2 Protein-Protein Interaction.
저자
by
Begnini, Fabio
;
Geschwindner, Stefan
;
Johansson, Patrik
;
Wissler, Lisa
;
Lewis, Richard J.
, et al.
소스
Journal of Medicinal Chemistry; 2/24/2022, Vol. 65 Issue 4, p3473-3517, 45p
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7 . Academic Journal
Biosensor-Enabled Deconvolution of the Avidity-Induced Affinity Enhancement for the SARS-CoV-2 Spike Protein and ACE2 Interaction.
저자
by
Gutgsell, Aspen Rene
;
Gunnarsson, Anders
;
Forssén, Patrik
;
Gordon, Euan
;
Fornstedt, Torgny
, et al.
소스
Analytical Chemistry; 1/18/2022, Vol. 94 Issue 2, p1187-1194, 8p
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7 . Academic Journal
Mining Natural Products for Macrocycles to Drug Difficult Targets.
저자
by
Begnini, Fabio
;
Poongavanam, Vasanthanathan
;
Over, Björn
;
Castaldo, Marie
;
Geschwindner, Stefan
, et al.
소스
Journal of Medicinal Chemistry; 1/28/2021, Vol. 64 Issue 2, p1054-1072, 19p
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7 . Academic Journal
Protease-activated receptor-2 ligands reveal orthosteric and allosteric mechanisms of receptor inhibition.
저자
by
Kennedy, Amanda J.
;
Sundström, Linda
;
Geschwindner, Stefan
;
Poon, Eunice K. Y.
;
Jiang, Yuhong
, et al.
소스
Communications Biology
. 12/17/2020, Vol. 3 Issue 1, p1-13. 13p.
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7 . Academic Journal
Synthesis and structure-activity relationship of 4-(1,3-benzothiazol-2-yl)-thiophene-2-sulfonamides as cyclin-dependent kinase 5 (cdk5)/p25 inhibitors
저자
by
Malmström, Jonas
;
Viklund, Jenny
;
Slivo, Can
;
Costa, Ana
;
Maudet, Mickaël
, et al.
소스
In
Bioorganic & Medicinal Chemistry Letters
15 September 2012 22(18):5919-5923
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