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1 . Academic Journal
A virtual library of small molecules mimicking dipeptides.
저자
by
Lim, Victor Jun Yu
;
Gerber, Hans‐Dieter
;
Schihada, Hannes
;
Trinh, Van Tuan
;
Hilger, Daniel
, et al.
소스
Archiv der Pharmazie; May2024, Vol. 357 Issue 5, p1-13, 13p
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7 . Academic Journal
Facile synthesis of substituted 2,3,4,7-tetrahydro-1 H-azepines via ring-closing metathesis
저자
by
Brass, Sascha
;
Gerber, Hans-Dieter
;
Dörr, Stefanie
;
Diederich, Wibke E.
.
소스
In
Tetrahedron
2006 62(8):1777-1786
Full Text (ScienceDirect)
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6 . Academic Journal
Structural and Biochemical Investigation of the Heterodimeric Murine tRNA-Guanine Transglycosylase.
저자
by
Sebastiani, Maurice
;
Behrens, Christina
;
Dörr, Stefanie
;
Gerber, Hans-Dieter
;
Benazza, Rania
, et al.
소스
ACS Chemical Biology; 8/19/2022, Vol. 17 Issue 8, p2229-2247, 19p
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7 . Academic Journal
Frag4Lead: growing crystallographic fragment hits by catalog using fragment‐guided template docking.
저자
by
Metz, Alexander
;
Wollenhaupt, Jan
;
Glöckner, Steffen
;
Messini, Niki
;
Huber, Simon
, et al.
소스
Acta Crystallographica: Section D, Structural Biology
. Sep2021, Vol. 77 Issue 9, p1168-1182. 15p.
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7 . Academic Journal
Surprising Non-Additivity of Methyl Groups in Drug–Kinase Interaction.
저자
by
Wienen-Schmidt, Barbara
;
Schmidt, Denis
;
Gerber, Hans-Dieter
;
Heine, Andreas
;
Gohlke, Holger
, et al.
소스
ACS Chemical Biology; Dec2019, Vol. 14 Issue 12, p2585-2594, 10p
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7 . Academic Journal
Paradoxically, Most Flexible Ligand Binds Most Entropy-Favored: Intriguing Impact of Ligand Flexibility and Solvation on Drug–Kinase Binding.
저자
by
Wienen-Schmidt, Barbara
;
Jonker, Hendrik R. A.
;
Wulsdorf, Tobias
;
Gerber, Hans-Dieter
;
Saxena, Krishna
, et al.
소스
Journal of Medicinal Chemistry; 7/15/2018, Vol. 61 Issue 14, p5922-5933, 12p
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7 . Academic Journal
Charges Shift Protonation: Neutron Diffraction Reveals that Aniline and 2-Aminopyridine Become Protonated Upon Binding to Trypsin.
저자
by
Schiebel, Johannes
;
Gaspari, Roberto
;
Sandner, Anna
;
Ngo, Khang
;
Gerber, Hans‐Dieter
, et al.
소스
Angewandte Chemie International Edition
. 4/18/2017, Vol. 56 Issue 17, p4887-4890. 4p.
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7 . Academic Journal
Kinetic and Structural Insights into the Mechanism of Binding of Sulfonamides to Human Carbonic Anhydrase by Computational and Experimental Studies.
저자
by
Gaspari, Roberto
;
Rechlin, Chris
;
Heine, Andreas
;
Bottegoni, Giovanni
;
Rocchia, Walter
, et al.
소스
Journal of Medicinal Chemistry
. 5/12/2016, Vol. 59 Issue 9, p4245-4256. 12p.
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7 . Academic Journal
Frontiers in Medicinal Chemistry 2015: Meet the Experts of MedChem near the Cradle of Medicinal and Pharmaceutical Chemistry.
저자
by
Wegscheid‐Gerlach, Christof
;
Gerber, Hans‐Dieter
;
Diederich, Wibke E.
.
소스
ChemMedChem; Jul2015, Vol. 10 Issue 7, p1267-1271, 5p
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5 . Academic Journal
Investigation of Specificity Determinants in Bacterial tRNA-Guanine Transglycosylase Reveals Queuine, the Substrate of Its Eucaryotic Counterpart, as Inhibitor
저자
by
Biela, Inna
;
Tidten-Luksch, Naomi
;
Immekus, Florian
;
Glinca, Serghei
;
Nguyen, Tran Xuan Phong
, et al.
소스
PLoS ONE
. May2013, Vol. 8 Issue 5, p1-19. 19p.
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