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1 .
Nintedanib: From Discovery to the Clinic
저자
by
Claudia Dallinger
;
Frank Hilberg
;
Stefan-Lutz Wollin
;
Rudolf Binder
;
Gerald Juergen Roth
, et al.
소스
Journal of Medicinal Chemistry
. 58:1053-1063
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7 .
Discovery of BI-2545: A Novel Autotaxin Inhibitor That Significantly Reduces LPA Levels in Vivo
저자
by
Helmut Romig
;
Sandra Handschuh
;
Tom Bretschneider
;
Bernd Nosse
;
Marco Ferrara
, et al.
소스
ACS medicinal chemistry letters
. 8(12)
Open Access (OpenAIRE)
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7 .
Discovery and Development of Nintedanib: A Novel Antiangiogenic and Antifibrotic Agent
저자
by
Rozsa Schlenker-Herceg
;
Florian Colbatzky
;
Rolf Kaiser
;
Alexander Pautsch
;
Rudolf Binder
, et al.
소스
Successful Drug Discovery
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7 .
Design, Synthesis, and Evaluation of Indolinones as Inhibitors of the Transforming Growth Factor β Receptor I (TGFβRI)
저자
by
Patrick Baum
;
Trixi Brandl
;
Detlev Mennerich
;
Stefan Hoerer
;
Gisela Schnapp
, et al.
소스
Journal of Medicinal Chemistry
. 53:7287-7295
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7 .
Design, synthesis and evaluation of MCH receptor 1 antagonists--Part III: Discovery of pre-clinical development candidate BI 186908
저자
by
Thorsten Lehmann
;
Ralf Lotz
;
Thorsten Oost
;
Mueller Stephan Georg
;
Klaus Rudolf
, et al.
소스
Bioorganicmedicinal chemistry letters
. 25(16)
Full Text (ScienceDirect)
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7 .
Design, synthesis and evaluation of MCH receptor 1 antagonists--Part I: Optimization of HTS hits towards an in vivo efficacious tool compound BI 414
저자
by
Gerd-Michael Maier
;
Thorsten Lehmann
;
Ralf Lotz
;
Jörg Kley
;
Martin Lenter
, et al.
소스
Bioorganicmedicinal chemistry letters
. 25(16)
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7 .
Design, synthesis and evaluation of MCH receptor 1 antagonists--Part II: Optimization of pyridazines toward reduced phospholipidosis and hERG inhibition
저자
by
Kirsten Arndt
;
Ralf Lotz
;
Klaus Rudolf
;
Thorsten Lehmann
;
Mueller Stephan Georg
, et al.
소스
Bioorganicmedicinal chemistry letters
. 25(16)
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7 .
Growth inhibition and induction of apoptosis in acute myeloid leukemia cells by new indolinone derivatives targeting fibroblast growth factor, platelet-derived growth factor, and vascular endothelial growth factor receptors
저자
by
Björn Steffen
;
Astrid Kolkmeyer
;
Carsten Müller-Tidow
;
Emma Kulimova
;
Frank Hilberg
, et al.
소스
Molecular Cancer Therapeutics
. 5:3105-3112
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7 .
The Oncogenic TLS-ERG Fusion Protein Exerts Different Effects in Hematopoietic Cells and Fibroblasts
저자
by
Howard A. Chansky
;
Anna Zielinska-Kwiatkowska
;
Hsien-Ming Hu
;
Liu Yang
;
Gerald Juergen Roth
, et al.
소스
Molecular and Cellular Biology
. 25:6235-6246
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7 .
Platelet-Active Drugs: The Relationships Among Dose, Effectiveness, and Side Effects
저자
by
Jack Hirsh
;
Gerald Juergen Roth
;
Carlo Patrono
;
Barry S. Coller
;
Garret A. FitzGerald
.
소스
Chest
. 126:234S-264S
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